Assay Detail
Functional
CHEMBL1614276
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: uHTS luminescence assay for the identification of compounds that inhibit NOD2 in MDP treated cells. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1566, AID1579, AID1849, AID2260, AID2335, AID2469, AID2503, AID2800]
545
Total Activities
545
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 545 | 5.20 | 7.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1597561 | — | — | 1 | 7.44 |
| CHEMBL3194944 | — | — | 1 | 6.99 |
| CHEMBL3195322 | — | — | 1 | 6.63 |
| CHEMBL3210725 | — | — | 1 | 6.32 |
| CHEMBL1415184 | — | — | 1 | 6.21 |
| CHEMBL1439315 | — | — | 1 | 6.16 |
| CHEMBL1580556 | — | — | 1 | 6.06 |
| CHEMBL1507713 | — | — | 1 | 5.94 |
| CHEMBL1520241 | — | — | 1 | 5.93 |
| CHEMBL1502883 | — | — | 1 | 5.93 |
| CHEMBL1319304 | — | — | 1 | 5.90 |
| CHEMBL1538692 | — | — | 1 | 5.89 |
| CHEMBL1569174 | — | — | 1 | 5.89 |
| CHEMBL1505956 | — | — | 1 | 5.83 |
| CHEMBL1486619 | — | — | 1 | 5.76 |
| CHEMBL1466636 | — | — | 1 | 5.76 |
| CHEMBL1483975 | — | — | 1 | 5.75 |
| CHEMBL257286 | — | — | 1 | 5.74 |
| CHEMBL1306524 | — | — | 1 | 5.72 |
| CHEMBL1480238 | — | — | 1 | 5.72 |
| CHEMBL1332003 | — | — | 1 | 5.71 |
| CHEMBL1333821 | — | — | 1 | 5.71 |
| CHEMBL1372398 | — | — | 1 | 5.71 |
| CHEMBL578257 | — | — | 1 | 5.71 |
| CHEMBL1320669 | — | — | 1 | 5.69 |
| CHEMBL1424697 | — | — | 1 | 5.67 |
| CHEMBL2006780 | — | — | 1 | 5.67 |
| CHEMBL585502 | — | — | 1 | 5.66 |
| CHEMBL1305930 | — | — | 1 | 5.64 |
| CHEMBL1465720 | — | — | 1 | 5.63 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1597561 | — | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL3194944 | — | IC50 | = | 103.0 | nM | 6.99 |
| CHEMBL3195322 | — | IC50 | = | 233.0 | nM | 6.63 |
| CHEMBL3210725 | — | IC50 | = | 480.0 | nM | 6.32 |
| CHEMBL1415184 | — | IC50 | = | 609.0 | nM | 6.21 |
| CHEMBL1439315 | — | IC50 | = | 695.0 | nM | 6.16 |
| CHEMBL1580556 | — | IC50 | = | 875.0 | nM | 6.06 |
| CHEMBL1507713 | — | IC50 | = | 1146.0 | nM | 5.94 |
| CHEMBL1520241 | — | IC50 | = | 1182.0 | nM | 5.93 |
| CHEMBL1502883 | — | IC50 | = | 1184.0 | nM | 5.93 |
| CHEMBL1319304 | — | IC50 | = | 1270.0 | nM | 5.90 |
| CHEMBL1569174 | — | IC50 | = | 1301.0 | nM | 5.89 |
| CHEMBL1538692 | — | IC50 | = | 1273.0 | nM | 5.89 |
| CHEMBL1505956 | — | IC50 | = | 1471.0 | nM | 5.83 |
| CHEMBL1486619 | — | IC50 | = | 1728.0 | nM | 5.76 |
| CHEMBL1466636 | — | IC50 | = | 1738.0 | nM | 5.76 |
| CHEMBL1483975 | — | IC50 | = | 1761.0 | nM | 5.75 |
| CHEMBL257286 | — | IC50 | = | 1832.0 | nM | 5.74 |
| CHEMBL1480238 | — | IC50 | = | 1917.0 | nM | 5.72 |
| CHEMBL1306524 | — | IC50 | = | 1906.0 | nM | 5.72 |
| CHEMBL1372398 | — | IC50 | = | 1950.0 | nM | 5.71 |
| CHEMBL1333821 | — | IC50 | = | 1928.0 | nM | 5.71 |
| CHEMBL578257 | — | IC50 | = | 1947.0 | nM | 5.71 |
| CHEMBL1332003 | — | IC50 | = | 1960.0 | nM | 5.71 |
| CHEMBL1320669 | — | IC50 | = | 2054.0 | nM | 5.69 |
| CHEMBL2006780 | — | IC50 | = | 2112.0 | nM | 5.67 |
| CHEMBL1424697 | — | IC50 | = | 2140.0 | nM | 5.67 |
| CHEMBL585502 | — | IC50 | = | 2199.0 | nM | 5.66 |
| CHEMBL1305930 | — | IC50 | = | 2289.0 | nM | 5.64 |
| CHEMBL1465720 | — | IC50 | = | 2361.0 | nM | 5.63 |
| CHEMBL1565526 | — | IC50 | = | 2373.0 | nM | 5.62 |
| CHEMBL1610725 | — | IC50 | = | 2393.0 | nM | 5.62 |
| CHEMBL1589670 | — | IC50 | = | 2407.0 | nM | 5.62 |
| CHEMBL190346 | — | IC50 | = | 2390.0 | nM | 5.62 |
| CHEMBL578944 | — | IC50 | = | 2480.0 | nM | 5.61 |
| CHEMBL1361883 | — | IC50 | = | 2483.0 | nM | 5.61 |
| CHEMBL1455542 | — | IC50 | = | 2585.0 | nM | 5.59 |
| CHEMBL3199186 | — | IC50 | = | 2703.0 | nM | 5.57 |
| CHEMBL1504069 | — | IC50 | = | 2701.0 | nM | 5.57 |
| CHEMBL1337226 | — | IC50 | = | 2705.0 | nM | 5.57 |
| CHEMBL1531328 | — | IC50 | = | 2712.0 | nM | 5.57 |
| CHEMBL1451348 | — | IC50 | = | 2679.0 | nM | 5.57 |
| CHEMBL1301943 | — | IC50 | = | 2745.0 | nM | 5.56 |
| CHEMBL1414053 | — | IC50 | = | 2855.0 | nM | 5.54 |
| CHEMBL1346518 | — | IC50 | = | 2938.0 | nM | 5.53 |
| CHEMBL1583914 | — | IC50 | = | 2928.0 | nM | 5.53 |
| CHEMBL1525735 | — | IC50 | = | 2943.0 | nM | 5.53 |
| CHEMBL1324011 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL1486981 | — | IC50 | = | 3039.0 | nM | 5.52 |
| CHEMBL1468181 | — | IC50 | = | 3044.0 | nM | 5.52 |