Assay Detail
Functional
CHEMBL1614409
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence counterscreen assay for TRPN1 agonists: dose response cell-based high-throughput screening assay to identify agonists of the transient receptor potential channel ML3 (TRPML3). (Class of assay: confirmatory) [Related pubchem assays: 1424, 1448 ]
77
Total Activities
77
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 77 | 5.34 | 6.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1377193 | — | — | 1 | 6.54 |
| CHEMBL1414923 | — | — | 1 | 5.99 |
| CHEMBL1569585 | — | — | 1 | 5.95 |
| CHEMBL1352344 | — | — | 1 | 5.72 |
| CHEMBL1490716 | — | — | 1 | 5.61 |
| CHEMBL1527735 | — | — | 1 | 5.56 |
| CHEMBL1575416 | — | — | 1 | 5.40 |
| CHEMBL1543131 | — | — | 1 | 5.40 |
| CHEMBL1574121 | — | — | 1 | 5.35 |
| CHEMBL1348043 | — | — | 1 | 5.34 |
| CHEMBL1605435 | — | — | 1 | 5.28 |
| CHEMBL1402083 | — | — | 1 | 5.27 |
| CHEMBL1971695 | — | — | 1 | 5.23 |
| CHEMBL1494852 | — | — | 1 | 5.21 |
| CHEMBL1313434 | — | — | 1 | 5.10 |
| CHEMBL1504676 | — | — | 1 | 5.05 |
| CHEMBL1342776 | — | — | 1 | 4.97 |
| CHEMBL1586687 | — | — | 1 | 4.91 |
| CHEMBL3039775 | — | — | 1 | 4.85 |
| CHEMBL581449 | — | — | 1 | 4.83 |
| CHEMBL1329925 | — | — | 1 | 4.61 |
| CHEMBL1507439 | — | — | 1 | - |
| CHEMBL601135 | — | — | 1 | - |
| CHEMBL1603731 | — | — | 1 | - |
| CHEMBL1389483 | — | — | 1 | - |
| CHEMBL455399 | — | — | 1 | - |
| CHEMBL1484458 | — | — | 1 | - |
| CHEMBL1330018 | — | — | 1 | - |
| CHEMBL1428566 | — | — | 1 | - |
| CHEMBL3194037 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1377193 | — | EC50 | = | 292.0 | nM | 6.54 |
| CHEMBL1414923 | — | EC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL1569585 | — | EC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL1352344 | — | EC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1490716 | — | EC50 | = | 2430.0 | nM | 5.61 |
| CHEMBL1527735 | — | EC50 | = | 2760.0 | nM | 5.56 |
| CHEMBL1575416 | — | EC50 | = | 3960.0 | nM | 5.40 |
| CHEMBL1543131 | — | EC50 | = | 3970.0 | nM | 5.40 |
| CHEMBL1574121 | — | EC50 | = | 4500.0 | nM | 5.35 |
| CHEMBL1348043 | — | EC50 | = | 4560.0 | nM | 5.34 |
| CHEMBL1605435 | — | EC50 | = | 5210.0 | nM | 5.28 |
| CHEMBL1402083 | — | EC50 | = | 5420.0 | nM | 5.27 |
| CHEMBL1971695 | — | EC50 | = | 5890.0 | nM | 5.23 |
| CHEMBL1494852 | — | EC50 | = | 6230.0 | nM | 5.21 |
| CHEMBL1313434 | — | EC50 | = | 7930.0 | nM | 5.10 |
| CHEMBL1504676 | — | EC50 | = | 8880.0 | nM | 5.05 |
| CHEMBL1342776 | — | EC50 | = | 10700.0 | nM | 4.97 |
| CHEMBL1586687 | — | EC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL3039775 | — | EC50 | = | 14200.0 | nM | 4.85 |
| CHEMBL581449 | — | EC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL1329925 | — | EC50 | = | 24300.0 | nM | 4.61 |
| CHEMBL1602160 | — | EC50 | > | 9970.0 | nM | - |
| CHEMBL1430184 | — | EC50 | > | 9970.0 | nM | - |
| CHEMBL1393535 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1351173 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1509135 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1351659 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1446321 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1470369 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1408066 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1603040 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1383045 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1419072 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1516758 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1319502 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1429822 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1602153 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1588763 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1585420 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1994036 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1506427 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL3194037 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1428566 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1330018 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1484458 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL455399 | — | EC50 | > | 1110.0 | nM | - |
| CHEMBL1389483 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL1603731 | — | EC50 | > | 29900.0 | nM | - |
| CHEMBL601135 | — | EC50 | > | 3320.0 | nM | - |
| CHEMBL1507439 | — | EC50 | > | 29900.0 | nM | - |