Assay Detail
Functional
CHEMBL1614432
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response Confirmation for Calpain Inhibitors. (Class of assay: confirmatory) [Related pubchem assays: 1236 (Primary screen preceding this confirmatory assay.)]
1128
Total Activities
1127
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Sus scrofa |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1128 | 5.07 | 6.35 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1477723 | — | — | 1 | 6.35 |
| CHEMBL1347786 | — | — | 1 | 6.34 |
| CHEMBL1438899 | — | — | 1 | 6.29 |
| CHEMBL1539019 | — | — | 1 | 6.27 |
| CHEMBL1532819 | — | — | 1 | 6.22 |
| CHEMBL1521078 | — | — | 1 | 6.18 |
| CHEMBL1322699 | — | — | 1 | 6.17 |
| CHEMBL1583674 | — | — | 1 | 6.17 |
| CHEMBL1427748 | — | — | 1 | 6.14 |
| CHEMBL1482453 | — | — | 1 | 6.13 |
| CHEMBL1485525 | — | — | 1 | 6.13 |
| CHEMBL1528647 | — | — | 1 | 6.11 |
| CHEMBL1452872 | — | — | 1 | 6.10 |
| CHEMBL1531389 | — | — | 1 | 6.09 |
| CHEMBL1413854 | — | — | 1 | 6.05 |
| CHEMBL1299610 | — | — | 1 | 6.05 |
| CHEMBL1526819 | — | — | 1 | 6.04 |
| CHEMBL1448876 | — | — | 1 | 6.04 |
| CHEMBL1364493 | — | — | 1 | 6.04 |
| CHEMBL1366209 | — | — | 1 | 6.04 |
| CHEMBL1393609 | — | — | 1 | 6.03 |
| CHEMBL1439185 | — | — | 1 | 5.99 |
| CHEMBL1385264 | — | — | 1 | 5.98 |
| CHEMBL1385374 | — | — | 1 | 5.98 |
| CHEMBL1358863 | — | — | 1 | 5.96 |
| CHEMBL1504385 | — | — | 1 | 5.96 |
| CHEMBL1351983 | — | — | 1 | 5.96 |
| CHEMBL1382924 | — | — | 1 | 5.95 |
| CHEMBL1447492 | — | — | 1 | 5.93 |
| CHEMBL1373569 | — | — | 1 | 5.88 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1477723 | — | IC50 | = | 443.54 | nM | 6.35 |
| CHEMBL1347786 | — | IC50 | = | 454.08 | nM | 6.34 |
| CHEMBL1438899 | — | IC50 | = | 513.77 | nM | 6.29 |
| CHEMBL1539019 | — | IC50 | = | 535.41 | nM | 6.27 |
| CHEMBL1532819 | — | IC50 | = | 608.01 | nM | 6.22 |
| CHEMBL1521078 | — | IC50 | = | 654.67 | nM | 6.18 |
| CHEMBL1322699 | — | IC50 | = | 672.92 | nM | 6.17 |
| CHEMBL1583674 | — | IC50 | = | 668.41 | nM | 6.17 |
| CHEMBL1427748 | — | IC50 | = | 718.77 | nM | 6.14 |
| CHEMBL1482453 | — | IC50 | = | 733.54 | nM | 6.13 |
| CHEMBL1485525 | — | IC50 | = | 737.08 | nM | 6.13 |
| CHEMBL1528647 | — | IC50 | = | 777.01 | nM | 6.11 |
| CHEMBL1452872 | — | IC50 | = | 795.91 | nM | 6.10 |
| CHEMBL1531389 | — | IC50 | = | 802.92 | nM | 6.09 |
| CHEMBL1299610 | — | IC50 | = | 898.82 | nM | 6.05 |
| CHEMBL1413854 | — | IC50 | = | 894.94 | nM | 6.05 |
| CHEMBL1526819 | — | IC50 | = | 903.95 | nM | 6.04 |
| CHEMBL1364493 | — | IC50 | = | 909.97 | nM | 6.04 |
| CHEMBL1366209 | — | IC50 | = | 916.9 | nM | 6.04 |
| CHEMBL1448876 | — | IC50 | = | 916.92 | nM | 6.04 |
| CHEMBL1393609 | — | IC50 | = | 930.68 | nM | 6.03 |
| CHEMBL1439185 | — | IC50 | = | 1018.61 | nM | 5.99 |
| CHEMBL1385374 | — | IC50 | = | 1042.87 | nM | 5.98 |
| CHEMBL1385264 | — | IC50 | = | 1044.74 | nM | 5.98 |
| CHEMBL1351983 | — | IC50 | = | 1101.08 | nM | 5.96 |
| CHEMBL1504385 | — | IC50 | = | 1104.49 | nM | 5.96 |
| CHEMBL1358863 | — | IC50 | = | 1089.97 | nM | 5.96 |
| CHEMBL1382924 | — | IC50 | = | 1113.15 | nM | 5.95 |
| CHEMBL1447492 | — | IC50 | = | 1186.18 | nM | 5.93 |
| CHEMBL1373569 | — | IC50 | = | 1309.31 | nM | 5.88 |
| CHEMBL1606087 | — | IC50 | = | 1360.11 | nM | 5.87 |
| CHEMBL1346061 | — | IC50 | = | 1420.18 | nM | 5.85 |
| CHEMBL1518193 | — | IC50 | = | 1424.32 | nM | 5.85 |
| CHEMBL1382623 | — | IC50 | = | 1426.51 | nM | 5.85 |
| CHEMBL1414508 | — | IC50 | = | 1424.19 | nM | 5.85 |
| CHEMBL1483192 | — | IC50 | = | 1511.73 | nM | 5.82 |
| CHEMBL1584754 | — | IC50 | = | 1588.43 | nM | 5.80 |
| CHEMBL3198457 | — | IC50 | = | 1587.37 | nM | 5.80 |
| CHEMBL1433052 | — | IC50 | = | 1581.3 | nM | 5.80 |
| CHEMBL1378300 | — | IC50 | = | 1630.66 | nM | 5.79 |
| CHEMBL1305142 | — | IC50 | = | 1631.68 | nM | 5.79 |
| CHEMBL1446629 | — | IC50 | = | 1627.6 | nM | 5.79 |
| CHEMBL1542578 | — | IC50 | = | 1658.79 | nM | 5.78 |
| CHEMBL1404786 | — | IC50 | = | 1735.73 | nM | 5.76 |
| CHEMBL1429036 | — | IC50 | = | 1799.02 | nM | 5.75 |
| CHEMBL1506889 | — | IC50 | = | 1778.45 | nM | 5.75 |
| CHEMBL63440 | ALOXISTATIN | IC50 | = | 1774.2 | nM | 5.75 |
| CHEMBL1460334 | — | IC50 | = | 1820.49 | nM | 5.74 |
| CHEMBL1410479 | — | IC50 | = | 1819.64 | nM | 5.74 |
| CHEMBL1412113 | — | IC50 | = | 1876.82 | nM | 5.73 |