Assay Detail
Functional
CHEMBL1614460
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence-based dose response cell-based high-throughput screening assay for agonists of NPY-Y1. (Class of assay: confirmatory) [Related pubchem assays: 1697 (Screening assay (NPY-Y1 agonists).), 1359 (Screening assay (NPY-Y2 potentiators or agonists).), 1304 (Screening assay (NPY-Y1 potentiators or agonists).), 1704 (Screening assay (CNGC inhibitors).), 1791 (Summary AID.)]
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 23 | 4.92 | 5.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1411397 | — | — | 1 | 5.15 |
| CHEMBL1301994 | — | — | 1 | 5.14 |
| CHEMBL1572588 | — | — | 1 | 5.13 |
| CHEMBL1312767 | — | — | 1 | 5.01 |
| CHEMBL1538224 | — | — | 1 | 4.93 |
| CHEMBL1519588 | — | — | 1 | 4.87 |
| CHEMBL526034 | — | — | 1 | 4.83 |
| CHEMBL1567983 | — | — | 1 | 4.81 |
| CHEMBL1560379 | — | — | 1 | 4.73 |
| CHEMBL1465891 | — | — | 1 | 4.56 |
| CHEMBL1603946 | — | — | 1 | - |
| CHEMBL1538198 | — | — | 1 | - |
| CHEMBL1422262 | — | — | 1 | - |
| CHEMBL1383943 | — | — | 1 | - |
| CHEMBL1448647 | — | — | 1 | - |
| CHEMBL1376325 | — | — | 1 | - |
| CHEMBL1979957 | — | — | 1 | - |
| CHEMBL1482965 | — | — | 1 | - |
| CHEMBL1534392 | — | — | 1 | - |
| CHEMBL1986557 | — | — | 1 | - |
| CHEMBL1406003 | — | — | 1 | - |
| CHEMBL1471980 | — | — | 1 | - |
| CHEMBL1597558 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1411397 | — | EC50 | = | 7050.0 | nM | 5.15 |
| CHEMBL1301994 | — | EC50 | = | 7164.0 | nM | 5.14 |
| CHEMBL1572588 | — | EC50 | = | 7410.0 | nM | 5.13 |
| CHEMBL1312767 | — | EC50 | = | 9709.0 | nM | 5.01 |
| CHEMBL1538224 | — | EC50 | = | 11619.0 | nM | 4.93 |
| CHEMBL1519588 | — | EC50 | = | 13550.0 | nM | 4.87 |
| CHEMBL526034 | — | EC50 | = | 14724.0 | nM | 4.83 |
| CHEMBL1567983 | — | EC50 | = | 15631.0 | nM | 4.81 |
| CHEMBL1560379 | — | EC50 | = | 18494.0 | nM | 4.73 |
| CHEMBL1465891 | — | EC50 | = | 27316.0 | nM | 4.56 |
| CHEMBL1603946 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1538198 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1422262 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1383943 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1448647 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1376325 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1979957 | — | EC50 | > | 11810.0 | nM | - |
| CHEMBL1482965 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1534392 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1986557 | — | EC50 | > | 3937.0 | nM | - |
| CHEMBL1406003 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1471980 | — | EC50 | > | 35430.0 | nM | - |
| CHEMBL1597558 | — | EC50 | > | 35430.0 | nM | - |