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Assay Detail

CHEMBL1614520

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: Anti-Viral Drugs Against Arbovirus Infections, a Confirmatory Screen. (Class of assay: confirmatory)
191
Total Activities
191
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category confirmatory
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 191 4.73 6.97

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3213254 1 6.97
CHEMBL1390450 1 6.78
CHEMBL1528840 1 6.75
CHEMBL1499652 1 6.38
CHEMBL3209279 1 6.28
CHEMBL1507013 1 5.85
CHEMBL1429270 1 5.84
CHEMBL1559138 1 5.78
CHEMBL1417376 1 5.64
CHEMBL1500409 1 5.62
CHEMBL1331422 1 5.51
CHEMBL1391672 1 5.40
CHEMBL1382563 1 5.34
CHEMBL415324 TRANILAST 3.0 1 5.32
CHEMBL1369254 1 5.31
CHEMBL1583917 1 5.30
CHEMBL1545848 1 5.29
CHEMBL1610008 1 5.27
CHEMBL1349072 1 5.25
CHEMBL1505572 1 5.23
CHEMBL1562713 1 5.21
CHEMBL1364290 1 5.12
CHEMBL1524932 1 5.12
CHEMBL1441583 1 5.07
CHEMBL1422748 1 5.05
CHEMBL1334503 1 5.04
CHEMBL1583227 1 5.03
CHEMBL1407771 1 5.03
CHEMBL1562136 1 5.01
CHEMBL515914 AZARIBINE 4.0 1 5.01

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3213254 IC50 = 108.0 nM 6.97
CHEMBL1390450 IC50 = 165.0 nM 6.78
CHEMBL1528840 IC50 = 178.0 nM 6.75
CHEMBL1499652 IC50 = 416.0 nM 6.38
CHEMBL3209279 IC50 = 524.0 nM 6.28
CHEMBL1507013 IC50 = 1400.0 nM 5.85
CHEMBL1429270 IC50 = 1446.0 nM 5.84
CHEMBL1559138 IC50 = 1675.0 nM 5.78
CHEMBL1417376 IC50 = 2283.0 nM 5.64
CHEMBL1500409 IC50 = 2417.0 nM 5.62
CHEMBL1331422 IC50 = 3056.0 nM 5.51
CHEMBL1391672 IC50 = 4005.0 nM 5.40
CHEMBL1382563 IC50 = 4594.0 nM 5.34
CHEMBL415324 TRANILAST IC50 = 4784.0 nM 5.32
CHEMBL1369254 IC50 = 4901.0 nM 5.31
CHEMBL1583917 IC50 = 4996.0 nM 5.30
CHEMBL1545848 IC50 = 5085.0 nM 5.29
CHEMBL1610008 IC50 = 5325.0 nM 5.27
CHEMBL1349072 IC50 = 5600.0 nM 5.25
CHEMBL1505572 IC50 = 5922.0 nM 5.23
CHEMBL1562713 IC50 = 6236.0 nM 5.21
CHEMBL1524932 IC50 = 7618.0 nM 5.12
CHEMBL1364290 IC50 = 7634.0 nM 5.12
CHEMBL1441583 IC50 = 8569.0 nM 5.07
CHEMBL1422748 IC50 = 8923.0 nM 5.05
CHEMBL1334503 IC50 = 9142.0 nM 5.04
CHEMBL1583227 IC50 = 9420.0 nM 5.03
CHEMBL1407771 IC50 = 9371.0 nM 5.03
CHEMBL515914 AZARIBINE IC50 = 9792.0 nM 5.01
CHEMBL1562136 IC50 = 9675.0 nM 5.01
CHEMBL1301429 IC50 = 9980.0 nM 5.00
CHEMBL1462011 IC50 = 10074.0 nM 5.00
CHEMBL1414498 IC50 = 10299.0 nM 4.99
CHEMBL1457718 IC50 = 10621.0 nM 4.97
CHEMBL1547896 IC50 = 11089.0 nM 4.96
CHEMBL1420606 IC50 = 11061.0 nM 4.96
CHEMBL1388081 IC50 = 11008.0 nM 4.96
CHEMBL1516943 IC50 = 12110.0 nM 4.92
CHEMBL1354041 IC50 = 12179.0 nM 4.91
CHEMBL1612354 IC50 = 12952.0 nM 4.89
CHEMBL1380661 IC50 = 13125.0 nM 4.88
CHEMBL3196867 IC50 = 13171.0 nM 4.88
CHEMBL3192328 IC50 = 13335.0 nM 4.88
CHEMBL1304974 IC50 = 14110.0 nM 4.85
CHEMBL3191171 IC50 = 14543.0 nM 4.84
CHEMBL1585563 IC50 = 14405.0 nM 4.84
CHEMBL3199860 IC50 = 15516.0 nM 4.81
CHEMBL1533248 IC50 = 15547.0 nM 4.81
CHEMBL1373855 IC50 = 15564.0 nM 4.81
CHEMBL2001743 IC50 = 15639.0 nM 4.81