Assay Detail
Functional
CHEMBL1614525
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence-based counterscreen assay for S1P4 antagonists: Cell-based dose response high throughput screening assay to identify antagonists of the Sphingosine 1-Phosphate Receptor 1 (S1P1). (Class of assay: confirmatory) [Related pubchem assays: 1524 (Confirmation screen.), 1510 (Primary screen.)]
100
Total Activities
100
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 100 | 5.05 | 6.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1537489 | — | — | 1 | 6.18 |
| CHEMBL586135 | — | — | 1 | 6.12 |
| CHEMBL1485168 | — | — | 1 | 5.92 |
| CHEMBL1487635 | — | — | 1 | 5.85 |
| CHEMBL171699 | — | — | 1 | 5.71 |
| CHEMBL1595015 | — | — | 1 | 5.64 |
| CHEMBL1334062 | — | — | 1 | 5.63 |
| CHEMBL1364999 | — | — | 1 | 5.48 |
| CHEMBL1361821 | — | — | 1 | 5.47 |
| CHEMBL1419909 | — | — | 1 | 5.46 |
| CHEMBL579318 | — | — | 1 | 5.44 |
| CHEMBL1332881 | — | — | 1 | 5.43 |
| CHEMBL1340713 | — | — | 1 | 5.43 |
| CHEMBL2000517 | — | — | 1 | 5.37 |
| CHEMBL1543295 | — | — | 1 | 5.37 |
| CHEMBL1613578 | — | — | 1 | 5.35 |
| CHEMBL1344225 | — | — | 1 | 5.35 |
| CHEMBL1439384 | — | — | 1 | 5.33 |
| CHEMBL1503962 | — | — | 1 | 5.32 |
| CHEMBL51931 | 9,10-PHENANTHRENEQUINONE | — | 1 | 5.30 |
| CHEMBL518292 | ISOVELLERAL | — | 1 | 5.30 |
| CHEMBL1301125 | — | — | 1 | 5.27 |
| CHEMBL1337227 | — | — | 1 | 5.26 |
| CHEMBL1540682 | — | — | 1 | 5.24 |
| CHEMBL1585527 | — | — | 1 | 5.23 |
| CHEMBL1432251 | — | — | 1 | 5.21 |
| CHEMBL1412583 | — | — | 1 | 5.21 |
| CHEMBL1447306 | — | — | 1 | 5.17 |
| CHEMBL1979747 | — | — | 1 | 5.17 |
| CHEMBL1369594 | — | — | 1 | 5.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1537489 | — | IC50 | = | 662.0 | nM | 6.18 |
| CHEMBL586135 | — | IC50 | = | 764.0 | nM | 6.12 |
| CHEMBL1485168 | — | IC50 | = | 1188.0 | nM | 5.92 |
| CHEMBL1487635 | — | IC50 | = | 1418.0 | nM | 5.85 |
| CHEMBL171699 | — | IC50 | = | 1960.0 | nM | 5.71 |
| CHEMBL1595015 | — | IC50 | = | 2285.0 | nM | 5.64 |
| CHEMBL1334062 | — | IC50 | = | 2343.0 | nM | 5.63 |
| CHEMBL1364999 | — | IC50 | = | 3285.0 | nM | 5.48 |
| CHEMBL1361821 | — | IC50 | = | 3417.0 | nM | 5.47 |
| CHEMBL1419909 | — | IC50 | = | 3429.0 | nM | 5.46 |
| CHEMBL579318 | — | IC50 | = | 3655.0 | nM | 5.44 |
| CHEMBL1332881 | — | IC50 | = | 3723.0 | nM | 5.43 |
| CHEMBL1340713 | — | IC50 | = | 3741.0 | nM | 5.43 |
| CHEMBL1543295 | — | IC50 | = | 4287.0 | nM | 5.37 |
| CHEMBL2000517 | — | IC50 | = | 4232.0 | nM | 5.37 |
| CHEMBL1613578 | — | IC50 | = | 4463.0 | nM | 5.35 |
| CHEMBL1344225 | — | IC50 | = | 4455.0 | nM | 5.35 |
| CHEMBL1439384 | — | IC50 | = | 4732.0 | nM | 5.33 |
| CHEMBL1503962 | — | IC50 | = | 4763.0 | nM | 5.32 |
| CHEMBL51931 | 9,10-PHENANTHRENEQUINONE | IC50 | = | 5020.0 | nM | 5.30 |
| CHEMBL518292 | ISOVELLERAL | IC50 | = | 4962.0 | nM | 5.30 |
| CHEMBL1301125 | — | IC50 | = | 5390.0 | nM | 5.27 |
| CHEMBL1337227 | — | IC50 | = | 5509.0 | nM | 5.26 |
| CHEMBL1540682 | — | IC50 | = | 5763.0 | nM | 5.24 |
| CHEMBL1585527 | — | IC50 | = | 5926.0 | nM | 5.23 |
| CHEMBL1432251 | — | IC50 | = | 6212.0 | nM | 5.21 |
| CHEMBL1412583 | — | IC50 | = | 6099.0 | nM | 5.21 |
| CHEMBL1447306 | — | IC50 | = | 6832.0 | nM | 5.17 |
| CHEMBL1979747 | — | IC50 | = | 6778.0 | nM | 5.17 |
| CHEMBL1369594 | — | IC50 | = | 6770.0 | nM | 5.17 |
| CHEMBL1309232 | — | IC50 | = | 7068.0 | nM | 5.15 |
| CHEMBL1468847 | — | IC50 | = | 7276.0 | nM | 5.14 |
| CHEMBL213580 | — | IC50 | = | 7195.0 | nM | 5.14 |
| CHEMBL1385784 | — | IC50 | = | 7322.0 | nM | 5.13 |
| CHEMBL1521989 | — | IC50 | = | 7637.0 | nM | 5.12 |
| CHEMBL1999049 | — | IC50 | = | 7505.0 | nM | 5.12 |
| CHEMBL1334984 | — | IC50 | = | 7959.0 | nM | 5.10 |
| CHEMBL1369655 | — | IC50 | = | 8147.0 | nM | 5.09 |
| CHEMBL1540377 | — | IC50 | = | 8586.0 | nM | 5.07 |
| CHEMBL610198 | — | IC50 | = | 8706.0 | nM | 5.06 |
| CHEMBL1451470 | — | IC50 | = | 8814.0 | nM | 5.05 |
| CHEMBL1572001 | — | IC50 | = | 9035.0 | nM | 5.04 |
| CHEMBL1426792 | — | IC50 | = | 9374.0 | nM | 5.03 |
| CHEMBL1526855 | — | IC50 | = | 9504.0 | nM | 5.02 |
| CHEMBL1362503 | — | IC50 | = | 9768.0 | nM | 5.01 |
| CHEMBL1566808 | — | IC50 | = | 9725.0 | nM | 5.01 |
| CHEMBL1605956 | — | IC50 | = | 9766.0 | nM | 5.01 |
| CHEMBL1558021 | — | IC50 | = | 9927.0 | nM | 5.00 |
| CHEMBL1440300 | — | IC50 | = | 10270.0 | nM | 4.99 |
| CHEMBL1343392 | — | IC50 | = | 10610.0 | nM | 4.97 |