Assay Detail
Functional
CHEMBL1614550
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based HTS Dose Confirmation to Identify Inhibitors of of 5'UTR Stem-Loop Driven Alpha-Synuclein mRNA Translation in H4 Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays: 1813 (Primary HTS), 1827 (Project Summary)]
184
Total Activities
184
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 184 | 6.46 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1555935 | — | — | 1 | 8.40 |
| CHEMBL3192138 | — | — | 1 | 8.22 |
| CHEMBL61 | PODOFILOX | 4.0 | 1 | 8.10 |
| CHEMBL1376974 | — | — | 1 | 7.96 |
| CHEMBL1536981 | — | — | 1 | 7.89 |
| CHEMBL1562575 | — | — | 1 | 7.80 |
| CHEMBL1357620 | — | — | 1 | 7.68 |
| CHEMBL1751 | DIGOXIN | 4.0 | 1 | 7.52 |
| CHEMBL3185655 | — | — | 1 | 7.43 |
| CHEMBL1587117 | — | — | 1 | 7.42 |
| CHEMBL1453996 | — | — | 1 | 7.41 |
| CHEMBL1342336 | — | — | 1 | 7.40 |
| CHEMBL1537509 | — | — | 1 | 7.33 |
| CHEMBL1368103 | — | — | 1 | 7.33 |
| CHEMBL513000 | — | — | 1 | 7.28 |
| CHEMBL501867 | VINCRISTINE SULFATE | 4.0 | 1 | 7.26 |
| CHEMBL222863 | OUABAIN | -1.0 | 1 | 7.19 |
| CHEMBL1307091 | — | — | 1 | 7.16 |
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 7.16 |
| CHEMBL290077 | — | — | 1 | 7.16 |
| CHEMBL1987060 | — | — | 1 | 7.15 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | -1.0 | 1 | 7.14 |
| CHEMBL1595169 | — | — | 1 | 7.14 |
| CHEMBL1347346 | — | — | 1 | 7.14 |
| CHEMBL1355541 | — | — | 1 | 7.09 |
| CHEMBL312862 | DEMECOLCINE | 2.0 | 1 | 7.07 |
| CHEMBL1333930 | — | — | 1 | 7.05 |
| CHEMBL1884996 | — | — | 1 | 7.04 |
| CHEMBL3195389 | — | — | 1 | 7.00 |
| CHEMBL423192 | ANISOMYCIN | — | 1 | 6.98 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1555935 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL3192138 | — | EC50 | = | 6.0 | nM | 8.22 |
| CHEMBL61 | PODOFILOX | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL1376974 | — | EC50 | = | 11.0 | nM | 7.96 |
| CHEMBL1536981 | — | EC50 | = | 13.0 | nM | 7.89 |
| CHEMBL1562575 | — | EC50 | = | 16.0 | nM | 7.80 |
| CHEMBL1357620 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL1751 | DIGOXIN | EC50 | = | 30.0 | nM | 7.52 |
| CHEMBL3185655 | — | EC50 | = | 37.0 | nM | 7.43 |
| CHEMBL1587117 | — | EC50 | = | 38.0 | nM | 7.42 |
| CHEMBL1453996 | — | EC50 | = | 39.0 | nM | 7.41 |
| CHEMBL1342336 | — | EC50 | = | 40.0 | nM | 7.40 |
| CHEMBL1537509 | — | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL1368103 | — | EC50 | = | 47.0 | nM | 7.33 |
| CHEMBL513000 | — | EC50 | = | 52.0 | nM | 7.28 |
| CHEMBL501867 | VINCRISTINE SULFATE | EC50 | = | 55.0 | nM | 7.26 |
| CHEMBL222863 | OUABAIN | EC50 | = | 64.0 | nM | 7.19 |
| CHEMBL290077 | — | EC50 | = | 70.0 | nM | 7.16 |
| CHEMBL1307091 | — | EC50 | = | 70.0 | nM | 7.16 |
| CHEMBL428647 | PACLITAXEL | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL1987060 | — | EC50 | = | 71.0 | nM | 7.15 |
| CHEMBL486504 | N-ACETYLCOLCHINOL | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL1347346 | — | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL1595169 | — | EC50 | = | 73.0 | nM | 7.14 |
| CHEMBL1355541 | — | EC50 | = | 82.0 | nM | 7.09 |
| CHEMBL312862 | DEMECOLCINE | EC50 | = | 85.0 | nM | 7.07 |
| CHEMBL1333930 | — | EC50 | = | 90.0 | nM | 7.05 |
| CHEMBL1884996 | — | EC50 | = | 92.0 | nM | 7.04 |
| CHEMBL3195389 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL423192 | ANISOMYCIN | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL373137 | — | EC50 | = | 106.0 | nM | 6.97 |
| CHEMBL1473676 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL1537098 | — | EC50 | = | 113.0 | nM | 6.95 |
| CHEMBL1423192 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL1312738 | — | EC50 | = | 118.0 | nM | 6.93 |
| CHEMBL460601 | — | EC50 | = | 118.0 | nM | 6.93 |
| CHEMBL1495092 | — | EC50 | = | 123.0 | nM | 6.91 |
| CHEMBL1602385 | — | EC50 | = | 124.0 | nM | 6.91 |
| CHEMBL1323774 | — | EC50 | = | 128.0 | nM | 6.89 |
| CHEMBL1540099 | — | EC50 | = | 133.0 | nM | 6.88 |
| CHEMBL1372889 | — | EC50 | = | 139.0 | nM | 6.86 |
| CHEMBL579318 | — | EC50 | = | 145.0 | nM | 6.84 |
| CHEMBL1406361 | — | EC50 | = | 149.0 | nM | 6.83 |
| CHEMBL1384292 | — | EC50 | = | 151.0 | nM | 6.82 |
| CHEMBL1528660 | — | EC50 | = | 156.0 | nM | 6.81 |
| CHEMBL1316831 | — | EC50 | = | 157.0 | nM | 6.80 |
| CHEMBL1392142 | — | EC50 | = | 159.0 | nM | 6.80 |
| CHEMBL1521023 | — | EC50 | = | 161.0 | nM | 6.79 |
| CHEMBL1307769 | — | EC50 | = | 170.0 | nM | 6.77 |
| CHEMBL1483593 | — | EC50 | = | 179.0 | nM | 6.75 |