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Assay Detail

CHEMBL1633575

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against thymidine kinase positive Cowpox virus harboring deltacrmA lacZ infected in HFF after 48 hrs by beta-galactosidase assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cowpox virus
Confidence 1 — Organism
Curated By Autocuration

Target

Cowpox virus (CHEMBL612672)
Type ORGANISM
Organism Cowpox virus

Publication

Activities of certain 5-substituted 4'-thiopyrimidine nucleosides against orthopoxvirus infections.
Kern ER, Prichard MN, Quenelle DC, Keith KA, Tiwari KN, Maddry JA, Secrist JA.
Antimicrob Agents Chemother (2009) 53 : 572 -579
PubMed 19029322 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 5.86 7.20

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1631219 1 7.20
CHEMBL1257073 TECOVIRIMAT 4.0 1 5.75
CHEMBL788 IDOXURIDINE 4.0 1 5.66
CHEMBL5314375 CIDOFOVIR 4.0 1 4.82

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1631219 EC50 = 63.0 nM 7.20
CHEMBL1257073 TECOVIRIMAT EC50 = 1800.0 nM 5.75
CHEMBL788 IDOXURIDINE EC50 = 2200.0 nM 5.66
CHEMBL5314375 CIDOFOVIR EC50 = 15000.0 nM 4.82