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Assay Detail

CHEMBL1637002

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Functional
Antiviral activity against J2R gene deficient Vaccinia virus harboring VVTK::luc infected in HFF assessed as reduction of plaque formation after 3 days
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vaccinia virus
Confidence 1 — Organism
Curated By Autocuration

Target

Vaccinia virus (CHEMBL613493)
Type ORGANISM
Organism Vaccinia virus

Publication

Activities of certain 5-substituted 4'-thiopyrimidine nucleosides against orthopoxvirus infections.
Kern ER, Prichard MN, Quenelle DC, Keith KA, Tiwari KN, Maddry JA, Secrist JA.
Antimicrob Agents Chemother (2009) 53 : 572 -579
PubMed 19029322 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 5.57 6.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1631219 1 6.52
CHEMBL788 IDOXURIDINE 4.0 1 5.15
CHEMBL5314375 CIDOFOVIR 4.0 1 5.03
CHEMBL1257073 TECOVIRIMAT 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1631219 EC50 = 300.0 nM 6.52
CHEMBL788 IDOXURIDINE EC50 = 7100.0 nM 5.15
CHEMBL5314375 CIDOFOVIR EC50 = 9400.0 nM 5.03
CHEMBL1257073 TECOVIRIMAT EC50 - -