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Assay Detail

CHEMBL1645780

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human MT4 lymphocytes after 48 hrs by MTT assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type MT4
Confidence 1 — Organism
Curated By Autocuration

Target

MT4 (CHEMBL388)
Type CELL-LINE
Organism Homo sapiens

Publication

Efficient synthesis and biological evaluation of epiceanothic acid and related compounds.
Zhang P, Xu L, Qian K, Liu J, Zhang L, Lee KH, Sun H.
Bioorg Med Chem Lett (2011) 21 : 338 -341
PubMed 21123066 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.62 4.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL404519 BEVIRIMAT 2.0 1 4.82
CHEMBL1644817 EPICEANOTHIC ACID 1 4.41
CHEMBL23236 BETULIN 1 -
CHEMBL1644922 1 -
CHEMBL1644923 1 -
CHEMBL1644924 1 -
CHEMBL1644925 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL404519 BEVIRIMAT IC50 = 15200.0 nM 4.82
CHEMBL1644817 EPICEANOTHIC ACID IC50 = 38900.0 nM 4.41
CHEMBL23236 BETULIN IC50 - -
CHEMBL1644922 IC50 - -
CHEMBL1644923 IC50 - -
CHEMBL1644924 IC50 - -
CHEMBL1644925 IC50 - -