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Assay Detail

CHEMBL1646836

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against X4 tropic HIV1 NL4.3 infected in human MT4 cells expressing CD4 and CXCR4 assessed as inhibition of virus-induced cytopathicity
28
Total Activities
28
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human immunodeficiency virus 1
Cell Type MT4
Confidence 1 — Organism
Curated By Autocuration

Target

Human immunodeficiency virus 1 (CHEMBL378)
Type ORGANISM
Organism Human immunodeficiency virus 1

Publication

Synthesis and SAR of novel CXCR4 antagonists that are potent inhibitors of T tropic (X4) HIV-1 replication.
Skerlj R, Bridger G, McEachern E, Harwig C, Smith C, Wilson T, Veale D, Yee H, Crawford J, Skupinska K, Wauthy R, Yang W, Zhu Y, Bogucki D, Di Fluri M, Langille J, Huskens D, De Clercq E, Schols D.
Bioorg Med Chem Lett (2011) 21 : 262 -266
PubMed 21109432 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 28 7.47 9.51

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1644082 1 9.51
CHEMBL1644088 1 9.40
CHEMBL1644081 1 9.00
CHEMBL1644073 1 8.70
CHEMBL1644080 1 8.38
CHEMBL1644092 1 8.14
CHEMBL1644089 1 8.10
CHEMBL1644096 1 7.96
CHEMBL1644078 1 7.92
CHEMBL1644085 1 7.85
CHEMBL1644074 1 7.77
CHEMBL1644072 1 7.75
CHEMBL1644075 1 7.70
CHEMBL1093008 1 7.68
CHEMBL1644094 1 7.68
CHEMBL1644079 1 7.66
CHEMBL1644076 1 7.16
CHEMBL1644095 1 6.99
CHEMBL1644077 1 6.98
CHEMBL1644071 1 6.98
CHEMBL1644083 1 6.91
CHEMBL1644070 1 6.78
CHEMBL1644086 1 5.61
CHEMBL1644091 1 5.55
CHEMBL1644087 1 5.45
CHEMBL1644093 1 4.70
CHEMBL1644090 1 -
CHEMBL1644084 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1644082 IC50 = 0.31 nM 9.51
CHEMBL1644088 IC50 = 0.4 nM 9.40
CHEMBL1644081 IC50 = 0.99 nM 9.00
CHEMBL1644073 IC50 = 2.0 nM 8.70
CHEMBL1644080 IC50 = 4.2 nM 8.38
CHEMBL1644092 IC50 = 7.2 nM 8.14
CHEMBL1644089 IC50 = 8.0 nM 8.10
CHEMBL1644096 IC50 = 10.9 nM 7.96
CHEMBL1644078 IC50 = 12.0 nM 7.92
CHEMBL1644085 IC50 = 14.0 nM 7.85
CHEMBL1644074 IC50 = 17.0 nM 7.77
CHEMBL1644072 IC50 = 18.0 nM 7.75
CHEMBL1644075 IC50 = 20.0 nM 7.70
CHEMBL1093008 IC50 = 21.0 nM 7.68
CHEMBL1644094 IC50 = 21.0 nM 7.68
CHEMBL1644079 IC50 = 22.0 nM 7.66
CHEMBL1644076 IC50 = 69.0 nM 7.16
CHEMBL1644095 IC50 = 103.0 nM 6.99
CHEMBL1644077 IC50 = 105.0 nM 6.98
CHEMBL1644071 IC50 = 104.0 nM 6.98
CHEMBL1644083 IC50 = 124.0 nM 6.91
CHEMBL1644070 IC50 = 165.0 nM 6.78
CHEMBL1644086 IC50 = 2480.0 nM 5.61
CHEMBL1644091 IC50 = 2830.0 nM 5.55
CHEMBL1644087 IC50 = 3570.0 nM 5.45
CHEMBL1644093 IC50 = 20100.0 nM 4.70
CHEMBL1644090 IC50 > 1160.0 nM -
CHEMBL1644084 IC50 > 1230.0 nM -