Assay Detail
Functional
CHEMBL1737862
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR analysis of SUMOylation using HTRF in an in-Vitro dose response assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2006, AID2011, AID2018, AID2069, AID2658]
113
Total Activities
109
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 113 | 4.94 | 5.71 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1518374 | — | — | 1 | 5.71 |
| CHEMBL1535613 | — | — | 1 | 5.70 |
| CHEMBL1713480 | — | — | 1 | 5.69 |
| CHEMBL1719957 | — | — | 1 | 5.66 |
| CHEMBL1736753 | — | — | 1 | 5.65 |
| CHEMBL1721038 | — | — | 1 | 5.62 |
| CHEMBL1703530 | — | — | 1 | 5.60 |
| CHEMBL1736986 | — | — | 1 | 5.60 |
| CHEMBL1727351 | — | — | 1 | 5.58 |
| CHEMBL1399979 | — | — | 1 | 5.58 |
| CHEMBL1507308 | — | — | 1 | 5.58 |
| CHEMBL1530437 | — | — | 1 | 5.57 |
| CHEMBL1731605 | — | — | 2 | 5.55 |
| CHEMBL1703238 | — | — | 1 | 5.47 |
| CHEMBL1722076 | — | — | 1 | 5.42 |
| CHEMBL1711163 | — | — | 1 | 5.42 |
| CHEMBL1706750 | — | — | 1 | 5.40 |
| CHEMBL1518888 | — | — | 1 | 5.39 |
| CHEMBL1518098 | — | — | 1 | 5.38 |
| CHEMBL1405964 | — | — | 1 | 5.38 |
| CHEMBL1612112 | — | — | 1 | 5.37 |
| CHEMBL1704267 | — | — | 2 | 5.36 |
| CHEMBL1720079 | — | — | 1 | 5.33 |
| CHEMBL1722739 | — | — | 1 | 5.33 |
| CHEMBL1446655 | — | — | 1 | 5.30 |
| CHEMBL1714309 | — | — | 1 | 5.29 |
| CHEMBL1328773 | — | — | 1 | 5.28 |
| CHEMBL1361703 | — | — | 1 | 5.24 |
| CHEMBL1732031 | — | — | 1 | 5.22 |
| CHEMBL1727199 | — | — | 1 | 5.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1518374 | — | IC50 | = | 1930.0 | nM | 5.71 |
| CHEMBL1535613 | — | IC50 | = | 2010.0 | nM | 5.70 |
| CHEMBL1713480 | — | IC50 | = | 2060.0 | nM | 5.69 |
| CHEMBL1719957 | — | IC50 | = | 2180.0 | nM | 5.66 |
| CHEMBL1736753 | — | IC50 | = | 2230.0 | nM | 5.65 |
| CHEMBL1721038 | — | IC50 | = | 2410.0 | nM | 5.62 |
| CHEMBL1736986 | — | IC50 | = | 2490.0 | nM | 5.60 |
| CHEMBL1703530 | — | IC50 | = | 2510.0 | nM | 5.60 |
| CHEMBL1727351 | — | IC50 | = | 2610.0 | nM | 5.58 |
| CHEMBL1399979 | — | IC50 | = | 2660.0 | nM | 5.58 |
| CHEMBL1507308 | — | IC50 | = | 2630.0 | nM | 5.58 |
| CHEMBL1530437 | — | IC50 | = | 2710.0 | nM | 5.57 |
| CHEMBL1731605 | — | IC50 | = | 2840.0 | nM | 5.55 |
| CHEMBL1703238 | — | IC50 | = | 3370.0 | nM | 5.47 |
| CHEMBL1722076 | — | IC50 | = | 3830.0 | nM | 5.42 |
| CHEMBL1711163 | — | IC50 | = | 3760.0 | nM | 5.42 |
| CHEMBL1706750 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL1518888 | — | IC50 | = | 4070.0 | nM | 5.39 |
| CHEMBL1405964 | — | IC50 | = | 4200.0 | nM | 5.38 |
| CHEMBL1518098 | — | IC50 | = | 4120.0 | nM | 5.38 |
| CHEMBL1612112 | — | IC50 | = | 4290.0 | nM | 5.37 |
| CHEMBL1704267 | — | IC50 | = | 4330.0 | nM | 5.36 |
| CHEMBL1731605 | — | IC50 | = | 4460.0 | nM | 5.35 |
| CHEMBL1720079 | — | IC50 | = | 4640.0 | nM | 5.33 |
| CHEMBL1722739 | — | IC50 | = | 4630.0 | nM | 5.33 |
| CHEMBL1446655 | — | IC50 | = | 4980.0 | nM | 5.30 |
| CHEMBL1714309 | — | IC50 | = | 5120.0 | nM | 5.29 |
| CHEMBL1328773 | — | IC50 | = | 5240.0 | nM | 5.28 |
| CHEMBL1361703 | — | IC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL1732031 | — | IC50 | = | 6040.0 | nM | 5.22 |
| CHEMBL1727199 | — | IC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL1562713 | — | IC50 | = | 6110.0 | nM | 5.21 |
| CHEMBL1402456 | — | IC50 | = | 6320.0 | nM | 5.20 |
| CHEMBL1728000 | — | IC50 | = | 6500.0 | nM | 5.19 |
| CHEMBL1308068 | — | IC50 | = | 6590.0 | nM | 5.18 |
| CHEMBL1706577 | — | IC50 | = | 7160.0 | nM | 5.14 |
| CHEMBL1706851 | — | IC50 | = | 7680.0 | nM | 5.12 |
| CHEMBL1704267 | — | IC50 | = | 8060.0 | nM | 5.09 |
| CHEMBL1706577 | — | IC50 | = | 9070.0 | nM | 5.04 |
| CHEMBL1727666 | — | IC50 | = | 9450.0 | nM | 5.03 |
| CHEMBL1575869 | — | IC50 | = | 10900.0 | nM | 4.96 |
| CHEMBL1519689 | — | IC50 | = | 11300.0 | nM | 4.95 |
| CHEMBL1728939 | — | IC50 | = | 11500.0 | nM | 4.94 |
| CHEMBL1372651 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL1502820 | — | IC50 | = | 12500.0 | nM | 4.90 |
| CHEMBL1725449 | — | IC50 | = | 12900.0 | nM | 4.89 |
| CHEMBL1302463 | — | IC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL1698818 | — | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL1715245 | — | IC50 | = | 14700.0 | nM | 4.83 |
| CHEMBL1706280 | — | IC50 | = | 16000.0 | nM | 4.80 |