Assay Detail
Binding
CHEMBL1738103
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for procaspase-3 activators: absorbance-based biochemical high throughput dose response assay for activators of procaspase-7. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID463141, AID463197, AID463210, AID488941, AID488954, AID493114, AID493115, AID504328, AID504330]
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 25 | 4.85 | 5.02 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1534294 | — | — | 1 | 5.02 |
| CHEMBL41286 | DIACEREIN | 3.0 | 1 | 4.83 |
| CHEMBL1603488 | — | — | 1 | 4.70 |
| CHEMBL1389713 | — | — | 1 | - |
| CHEMBL1504407 | — | — | 1 | - |
| CHEMBL1494574 | — | — | 1 | - |
| CHEMBL1299990 | — | — | 1 | - |
| CHEMBL1974856 | — | — | 1 | - |
| CHEMBL1585831 | — | — | 1 | - |
| CHEMBL1377382 | — | — | 1 | - |
| CHEMBL1358403 | — | — | 1 | - |
| CHEMBL1509137 | — | — | 1 | - |
| CHEMBL3191201 | — | — | 1 | - |
| CHEMBL1608043 | — | — | 1 | - |
| CHEMBL1404887 | — | — | 1 | - |
| CHEMBL1365411 | — | — | 1 | - |
| CHEMBL3192911 | — | — | 1 | - |
| CHEMBL3195241 | — | — | 1 | - |
| CHEMBL3195767 | — | — | 1 | - |
| CHEMBL1715943 | — | — | 1 | - |
| CHEMBL1490564 | — | — | 1 | - |
| CHEMBL1584696 | — | — | 1 | - |
| CHEMBL2004978 | — | — | 1 | - |
| CHEMBL1490809 | — | — | 1 | - |
| CHEMBL1470280 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1534294 | — | EC50 | = | 9486.0 | nM | 5.02 |
| CHEMBL41286 | DIACEREIN | EC50 | = | 14802.0 | nM | 4.83 |
| CHEMBL1603488 | — | EC50 | = | 20198.0 | nM | 4.70 |
| CHEMBL1389713 | — | EC50 | > | 85267.0 | nM | - |
| CHEMBL1504407 | — | EC50 | > | 85301.0 | nM | - |
| CHEMBL1494574 | — | EC50 | > | 85275.0 | nM | - |
| CHEMBL1299990 | — | EC50 | > | 85247.0 | nM | - |
| CHEMBL1974856 | — | EC50 | > | 85267.0 | nM | - |
| CHEMBL1585831 | — | EC50 | > | 85275.0 | nM | - |
| CHEMBL1377382 | — | EC50 | > | 85245.0 | nM | - |
| CHEMBL1358403 | — | EC50 | > | 85239.0 | nM | - |
| CHEMBL1509137 | — | EC50 | > | 85275.0 | nM | - |
| CHEMBL3191201 | — | EC50 | > | 85267.0 | nM | - |
| CHEMBL1608043 | — | EC50 | > | 85212.0 | nM | - |
| CHEMBL1404887 | — | EC50 | > | 85247.0 | nM | - |
| CHEMBL1365411 | — | EC50 | > | 85301.0 | nM | - |
| CHEMBL3192911 | — | EC50 | > | 3157.0 | nM | - |
| CHEMBL3195241 | — | EC50 | > | 85267.0 | nM | - |
| CHEMBL3195767 | — | EC50 | > | 85267.0 | nM | - |
| CHEMBL1715943 | — | EC50 | > | 85222.0 | nM | - |
| CHEMBL1490564 | — | EC50 | > | 85222.0 | nM | - |
| CHEMBL1584696 | — | EC50 | > | 85245.0 | nM | - |
| CHEMBL2004978 | — | EC50 | > | 85267.0 | nM | - |
| CHEMBL1490809 | — | EC50 | > | 85251.0 | nM | - |
| CHEMBL1470280 | — | EC50 | > | 85267.0 | nM | - |