Assay Detail
Functional
CHEMBL1738314
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 3. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2058, AID2079]
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 4.96 | 5.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1720530 | — | — | 1 | 5.18 |
| CHEMBL1708510 | — | — | 1 | 5.04 |
| CHEMBL1709028 | — | — | 1 | 4.82 |
| CHEMBL1727267 | — | — | 1 | 4.79 |
| CHEMBL1718866 | — | — | 1 | - |
| CHEMBL1709632 | — | — | 1 | - |
| CHEMBL1700099 | — | — | 1 | - |
| CHEMBL1700467 | — | — | 1 | - |
| CHEMBL1701030 | — | — | 1 | - |
| CHEMBL1723238 | — | — | 1 | - |
| CHEMBL1723578 | — | — | 1 | - |
| CHEMBL1704074 | — | — | 1 | - |
| CHEMBL1734603 | — | — | 1 | - |
| CHEMBL1716874 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1720530 | — | IC50 | = | 6580.0 | nM | 5.18 |
| CHEMBL1708510 | — | IC50 | = | 9080.0 | nM | 5.04 |
| CHEMBL1709028 | — | IC50 | = | 15100.0 | nM | 4.82 |
| CHEMBL1727267 | — | IC50 | = | 16400.0 | nM | 4.79 |
| CHEMBL1718866 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1709632 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1700099 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1700467 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1701030 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1723238 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1723578 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1704074 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1734603 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1716874 | — | IC50 | > | 32000.0 | nM | - |