Assay Detail
Functional
CHEMBL1738352
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PUBCHEM_BIOASSAY: Dose Response confirmation of Inhibitors of Mdm2/MdmX interaction using a Full-Length Luciferase Counterscreen assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID485346, AID488776]
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 5.38 | 6.86 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1579258 | — | — | 1 | 6.86 |
| CHEMBL3189193 | — | — | 1 | 5.80 |
| CHEMBL1370413 | — | — | 1 | 5.76 |
| CHEMBL48310 | HINOKITIOL | — | 1 | 5.64 |
| CHEMBL1352521 | — | — | 1 | 5.62 |
| CHEMBL1547940 | — | — | 1 | 5.62 |
| CHEMBL270605 | — | — | 1 | 5.57 |
| CHEMBL1603457 | — | — | 1 | 5.45 |
| CHEMBL1522344 | — | — | 1 | 5.41 |
| CHEMBL1536628 | — | — | 1 | 5.29 |
| CHEMBL1723414 | — | — | 1 | 5.24 |
| CHEMBL1538187 | — | — | 1 | 5.21 |
| CHEMBL1332955 | — | — | 1 | 5.13 |
| CHEMBL1459746 | — | — | 1 | 5.12 |
| CHEMBL1342054 | — | — | 1 | 5.05 |
| CHEMBL3197778 | — | — | 1 | 4.94 |
| CHEMBL1610180 | — | — | 1 | 4.90 |
| CHEMBL532504 | — | — | 1 | 4.86 |
| CHEMBL1342070 | — | — | 1 | 4.81 |
| CHEMBL601180 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1579258 | — | IC50 | = | 137.0 | nM | 6.86 |
| CHEMBL3189193 | — | IC50 | = | 1568.0 | nM | 5.80 |
| CHEMBL1370413 | — | IC50 | = | 1751.0 | nM | 5.76 |
| CHEMBL48310 | HINOKITIOL | IC50 | = | 2267.0 | nM | 5.64 |
| CHEMBL1352521 | — | IC50 | = | 2375.0 | nM | 5.62 |
| CHEMBL1547940 | — | IC50 | = | 2410.0 | nM | 5.62 |
| CHEMBL270605 | — | IC50 | = | 2671.0 | nM | 5.57 |
| CHEMBL1603457 | — | IC50 | = | 3582.0 | nM | 5.45 |
| CHEMBL1522344 | — | IC50 | = | 3869.0 | nM | 5.41 |
| CHEMBL1536628 | — | IC50 | = | 5162.0 | nM | 5.29 |
| CHEMBL1723414 | — | IC50 | = | 5780.0 | nM | 5.24 |
| CHEMBL1538187 | — | IC50 | = | 6227.0 | nM | 5.21 |
| CHEMBL1332955 | — | IC50 | = | 7439.0 | nM | 5.13 |
| CHEMBL1459746 | — | IC50 | = | 7639.0 | nM | 5.12 |
| CHEMBL1342054 | — | IC50 | = | 8880.0 | nM | 5.05 |
| CHEMBL3197778 | — | IC50 | = | 11478.0 | nM | 4.94 |
| CHEMBL1610180 | — | IC50 | = | 12535.0 | nM | 4.90 |
| CHEMBL532504 | — | IC50 | = | 13781.0 | nM | 4.86 |
| CHEMBL1342070 | — | IC50 | = | 15465.0 | nM | 4.81 |
| CHEMBL601180 | — | IC50 | > | 79000.0 | nM | - |