Assay Detail
Functional
CHEMBL1738365
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2013, AID2026]
38
Total Activities
38
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 38 | 6.07 | 6.90 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL394883 | — | — | 1 | 6.90 |
| CHEMBL1310336 | — | — | 1 | 6.87 |
| CHEMBL1484306 | — | — | 1 | 6.47 |
| CHEMBL1441155 | — | — | 1 | 6.45 |
| CHEMBL1578189 | — | — | 1 | 6.39 |
| CHEMBL1354041 | — | — | 1 | 6.38 |
| CHEMBL1567371 | — | — | 1 | 6.34 |
| CHEMBL1452959 | — | — | 1 | 6.30 |
| CHEMBL1421591 | — | — | 1 | 6.24 |
| CHEMBL1402920 | — | — | 1 | 6.15 |
| CHEMBL1507172 | — | — | 1 | 6.15 |
| CHEMBL1542168 | — | — | 1 | 6.12 |
| CHEMBL1431310 | — | — | 1 | 6.08 |
| CHEMBL1549881 | — | — | 1 | 6.07 |
| CHEMBL1420151 | — | — | 1 | 6.06 |
| CHEMBL1507657 | — | — | 1 | 6.06 |
| CHEMBL1431953 | — | — | 1 | 6.05 |
| CHEMBL1613157 | — | — | 1 | 6.04 |
| CHEMBL1582765 | — | — | 1 | 6.03 |
| CHEMBL1468612 | — | — | 1 | 6.02 |
| CHEMBL1411212 | — | — | 1 | 6.01 |
| CHEMBL1410009 | — | — | 1 | 6.01 |
| CHEMBL1445966 | — | — | 1 | 6.00 |
| CHEMBL1498988 | — | — | 1 | 6.00 |
| CHEMBL1460039 | — | — | 1 | 5.97 |
| CHEMBL1366039 | — | — | 1 | 5.97 |
| CHEMBL1575373 | — | — | 1 | 5.96 |
| CHEMBL1466203 | — | — | 1 | 5.94 |
| CHEMBL1464477 | — | — | 1 | 5.91 |
| CHEMBL1429129 | — | — | 1 | 5.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL394883 | — | IC50 | = | 125.0 | nM | 6.90 |
| CHEMBL1310336 | — | IC50 | = | 136.0 | nM | 6.87 |
| CHEMBL1484306 | — | IC50 | = | 342.0 | nM | 6.47 |
| CHEMBL1441155 | — | IC50 | = | 354.0 | nM | 6.45 |
| CHEMBL1578189 | — | IC50 | = | 407.0 | nM | 6.39 |
| CHEMBL1354041 | — | IC50 | = | 422.0 | nM | 6.38 |
| CHEMBL1567371 | — | IC50 | = | 457.0 | nM | 6.34 |
| CHEMBL1452959 | — | IC50 | = | 506.0 | nM | 6.30 |
| CHEMBL1421591 | — | IC50 | = | 577.0 | nM | 6.24 |
| CHEMBL1402920 | — | IC50 | = | 702.0 | nM | 6.15 |
| CHEMBL1507172 | — | IC50 | = | 709.0 | nM | 6.15 |
| CHEMBL1542168 | — | IC50 | = | 760.0 | nM | 6.12 |
| CHEMBL1431310 | — | IC50 | = | 831.0 | nM | 6.08 |
| CHEMBL1549881 | — | IC50 | = | 854.0 | nM | 6.07 |
| CHEMBL1507657 | — | IC50 | = | 865.0 | nM | 6.06 |
| CHEMBL1420151 | — | IC50 | = | 878.0 | nM | 6.06 |
| CHEMBL1431953 | — | IC50 | = | 893.0 | nM | 6.05 |
| CHEMBL1613157 | — | IC50 | = | 917.0 | nM | 6.04 |
| CHEMBL1582765 | — | IC50 | = | 928.0 | nM | 6.03 |
| CHEMBL1468612 | — | IC50 | = | 948.0 | nM | 6.02 |
| CHEMBL1410009 | — | IC50 | = | 978.0 | nM | 6.01 |
| CHEMBL1411212 | — | IC50 | = | 965.0 | nM | 6.01 |
| CHEMBL1445966 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1498988 | — | IC50 | = | 992.0 | nM | 6.00 |
| CHEMBL1460039 | — | IC50 | = | 1060.0 | nM | 5.97 |
| CHEMBL1366039 | — | IC50 | = | 1080.0 | nM | 5.97 |
| CHEMBL1575373 | — | IC50 | = | 1090.0 | nM | 5.96 |
| CHEMBL1466203 | — | IC50 | = | 1140.0 | nM | 5.94 |
| CHEMBL1464477 | — | IC50 | = | 1240.0 | nM | 5.91 |
| CHEMBL1429129 | — | IC50 | = | 1420.0 | nM | 5.85 |
| CHEMBL1420800 | — | IC50 | = | 1450.0 | nM | 5.84 |
| CHEMBL1448070 | — | IC50 | = | 1440.0 | nM | 5.84 |
| CHEMBL1386881 | — | IC50 | = | 1690.0 | nM | 5.77 |
| CHEMBL1545109 | — | IC50 | = | 1810.0 | nM | 5.74 |
| CHEMBL1611658 | — | IC50 | = | 1940.0 | nM | 5.71 |
| CHEMBL1546161 | — | IC50 | = | 2050.0 | nM | 5.69 |
| CHEMBL1572633 | — | IC50 | = | 2360.0 | nM | 5.63 |
| CHEMBL1581985 | — | IC50 | = | 2720.0 | nM | 5.57 |