Assay Detail
Unclassified
CHEMBL1738385
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Late stage results from the probe development effort to identify activators of signal transducer and activator of transcription 3 (STAT3). (Class of assay: screening) [Related pubchem assays (depositor defined):AID1267, AID1309, AID1318, AID1398, AID1406, AID1805, AID871, AID932] Panel member name: STAT3 Activation
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Unclassified |
| Category | screening |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Signal transducer and activator of transcription 3 (CHEMBL4026) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 14 | 7.07 | 8.98 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1389016 | — | — | 1 | 8.98 |
| CHEMBL1449962 | — | — | 1 | 8.66 |
| CHEMBL1703740 | — | — | 1 | 8.34 |
| CHEMBL1430610 | — | — | 1 | 8.09 |
| CHEMBL1729988 | — | — | 1 | 5.22 |
| CHEMBL1707774 | — | — | 1 | 5.16 |
| CHEMBL1722282 | — | — | 1 | 5.02 |
| CHEMBL1698563 | — | — | 1 | - |
| CHEMBL1701324 | — | — | 1 | - |
| CHEMBL1735352 | — | — | 1 | - |
| CHEMBL1717477 | — | — | 1 | - |
| CHEMBL1729319 | — | — | 1 | - |
| CHEMBL1736009 | — | — | 1 | - |
| CHEMBL1702219 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1389016 | — | EC50 | = | 1.04 | nM | 8.98 |
| CHEMBL1449962 | — | EC50 | = | 2.19 | nM | 8.66 |
| CHEMBL1703740 | — | EC50 | = | 4.55 | nM | 8.34 |
| CHEMBL1430610 | — | EC50 | = | 8.15 | nM | 8.09 |
| CHEMBL1729988 | — | EC50 | = | 6080.0 | nM | 5.22 |
| CHEMBL1707774 | — | EC50 | = | 6978.0 | nM | 5.16 |
| CHEMBL1722282 | — | EC50 | = | 9618.0 | nM | 5.02 |
| CHEMBL1698563 | — | EC50 | > | 5569.0 | nM | - |
| CHEMBL1701324 | — | EC50 | > | 55690.0 | nM | - |
| CHEMBL1735352 | — | EC50 | > | 55690.0 | nM | - |
| CHEMBL1717477 | — | EC50 | > | 55690.0 | nM | - |
| CHEMBL1729319 | — | EC50 | > | 5569.0 | nM | - |
| CHEMBL1736009 | — | EC50 | > | 5569.0 | nM | - |
| CHEMBL1702219 | — | EC50 | > | 55690.0 | nM | - |