Assay Detail
Functional
CHEMBL1738405
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: HTS Dose response counterscreen for assays utilizing the enzyme, beta-galactosidase - Set 3. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493098, AID493121, AID493159]
283
Total Activities
283
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Escherichia coli |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 283 | 4.42 | 4.78 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1522033 | — | — | 1 | 4.78 |
| CHEMBL2004847 | — | — | 1 | 4.48 |
| CHEMBL1610008 | — | — | 1 | 4.47 |
| CHEMBL3197091 | — | — | 1 | 4.44 |
| CHEMBL1533772 | — | — | 1 | 4.39 |
| CHEMBL355496 | — | — | 1 | 4.39 |
| CHEMBL1987894 | — | — | 1 | 4.38 |
| CHEMBL3191855 | — | — | 1 | 4.37 |
| CHEMBL1969046 | — | — | 1 | 4.36 |
| CHEMBL1733564 | — | — | 1 | 4.34 |
| CHEMBL1578670 | — | — | 1 | 4.33 |
| CHEMBL3196451 | — | — | 1 | 4.29 |
| CHEMBL1698464 | — | — | 1 | - |
| CHEMBL1324005 | — | — | 1 | - |
| CHEMBL1309432 | — | — | 1 | - |
| CHEMBL1717890 | — | — | 1 | - |
| CHEMBL1485865 | — | — | 1 | - |
| CHEMBL1965860 | — | — | 1 | - |
| CHEMBL3191691 | — | — | 1 | - |
| CHEMBL1965403 | — | — | 1 | - |
| CHEMBL387762 | — | — | 1 | - |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | — | 1 | - |
| CHEMBL1717415 | — | — | 1 | - |
| CHEMBL1447124 | — | — | 1 | - |
| CHEMBL1555566 | — | — | 1 | - |
| CHEMBL1467867 | — | — | 1 | - |
| CHEMBL1607475 | — | — | 1 | - |
| CHEMBL1587764 | — | — | 1 | - |
| CHEMBL1964407 | — | — | 1 | - |
| CHEMBL1342574 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1522033 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL2004847 | — | IC50 | = | 33000.0 | nM | 4.48 |
| CHEMBL1610008 | — | IC50 | = | 33800.0 | nM | 4.47 |
| CHEMBL3197091 | — | IC50 | = | 36100.0 | nM | 4.44 |
| CHEMBL1533772 | — | IC50 | = | 41000.0 | nM | 4.39 |
| CHEMBL355496 | — | IC50 | = | 40800.0 | nM | 4.39 |
| CHEMBL1987894 | — | IC50 | = | 41300.0 | nM | 4.38 |
| CHEMBL3191855 | — | IC50 | = | 43000.0 | nM | 4.37 |
| CHEMBL1969046 | — | IC50 | = | 43500.0 | nM | 4.36 |
| CHEMBL1733564 | — | IC50 | = | 46000.0 | nM | 4.34 |
| CHEMBL1578670 | — | IC50 | = | 46300.0 | nM | 4.33 |
| CHEMBL3196451 | — | IC50 | = | 50800.0 | nM | 4.29 |
| CHEMBL1431909 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1565536 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL393287 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL592124 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1704635 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL3192924 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1723955 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1733858 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1534949 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1312308 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1991431 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1424264 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1427185 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1487205 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1703076 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL3192555 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1462873 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1722738 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1458840 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1506256 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1997450 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL3191445 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL242163 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL212504 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1481383 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1338167 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1580684 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL2095095 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL3198396 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1470925 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1705093 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1463571 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1996730 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1527565 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1993788 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1734152 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1400481 | — | IC50 | > | 66600.0 | nM | - |
| CHEMBL1516474 | TEGASEROD MALEATE | IC50 | > | 66600.0 | nM | - |