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Compound Detail

CHEMBL1965860

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C/C(=N\NC(=S)NCCc1ccccc1)c1ccc(Cl)cc1Cl

Basic Information

ChEMBL ID CHEMBL1965860
Phase Preclinical
Structure Type MOL
InChI Key WRQPNTFOWSEHKM-CIAFOILYSA-N
4
Targets
4
Activities
2
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

366.3
MW (Da)
4.42
ALogP
2
HBA
2
HBD
36.4
PSA (Ų)
0.47
QED
0
Ro5 Violations
5
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C17H17Cl2N3S
MW 366.32
Aromatic Rings 2
Heavy Atoms 23
NP-Likeness -1.76

Activity Summary

EC50 3 meas. best 5.33
IC50 1 meas. best 4.82

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Streptococcus sp. 'group A'
CHEMBL612389
EC50 5.33 5.33 4656.0 1
Streptokinase A
CHEMBL1293228
EC50 5.18 5.18 6559.0 1
C-C chemokine receptor type 6
CHEMBL4423
IC50 4.82 4.82 15100.0 1
Streptococcus
CHEMBL612313
EC50 4.67 4.67 21245.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine