Assay Detail
Functional
CHEMBL1614538
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Response HTS to Identify Compounds Cytotoxic to Streptococcus. (Class of assay: confirmatory) [Related pubchem assays: 1900 (Counter Screen), 1677 (Project Summary), 1902 (Retest at Dose), 1662 (Primary HTS)]
3265
Total Activities
3262
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Streptococcus |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3265 | 5.06 | 7.19 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL586135 | — | — | 1 | 7.19 |
| CHEMBL529 | AZITHROMYCIN | 4.0 | 1 | 7.18 |
| CHEMBL1467058 | — | — | 1 | 7.15 |
| CHEMBL581257 | — | — | 1 | 7.07 |
| CHEMBL12131 | CLOSANTEL | 2.0 | 1 | 7.04 |
| CHEMBL1334646 | — | — | 1 | 7.01 |
| CHEMBL1444820 | — | — | 1 | 7.00 |
| CHEMBL1364011 | — | — | 1 | 6.97 |
| CHEMBL1537542 | — | — | 1 | 6.97 |
| CHEMBL1422253 | — | — | 1 | 6.96 |
| CHEMBL1485275 | — | — | 1 | 6.96 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | 4.0 | 1 | 6.96 |
| CHEMBL1382674 | — | — | 1 | 6.94 |
| CHEMBL1237072 | DIRITHROMYCIN | 4.0 | 1 | 6.93 |
| CHEMBL1318922 | — | — | 1 | 6.93 |
| CHEMBL1484438 | — | — | 1 | 6.91 |
| CHEMBL1516396 | — | — | 1 | 6.90 |
| CHEMBL1256686 | CALCIMYCIN | 2.0 | 1 | 6.89 |
| CHEMBL287542 | RAFOXANIDE | 2.0 | 1 | 6.86 |
| CHEMBL1528206 | — | — | 1 | 6.85 |
| CHEMBL278255 | CLINAFLOXACIN | 2.0 | 1 | 6.85 |
| CHEMBL1344339 | — | — | 1 | 6.83 |
| CHEMBL2146063 | CHLORTETRACYCLINE HYDROCHLORIDE | 4.0 | 1 | 6.83 |
| CHEMBL1342436 | — | — | 1 | 6.82 |
| CHEMBL1583292 | — | — | 1 | 6.78 |
| CHEMBL1385808 | — | — | 1 | 6.76 |
| CHEMBL1333965 | — | — | 1 | 6.74 |
| CHEMBL1545940 | — | — | 1 | 6.74 |
| CHEMBL1326397 | — | — | 1 | 6.64 |
| CHEMBL1493936 | — | — | 1 | 6.64 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL586135 | — | EC50 | = | 65.0 | nM | 7.19 |
| CHEMBL529 | AZITHROMYCIN | EC50 | = | 66.0 | nM | 7.18 |
| CHEMBL1467058 | — | EC50 | = | 71.0 | nM | 7.15 |
| CHEMBL581257 | — | EC50 | = | 85.0 | nM | 7.07 |
| CHEMBL12131 | CLOSANTEL | EC50 | = | 92.0 | nM | 7.04 |
| CHEMBL1334646 | — | EC50 | = | 98.0 | nM | 7.01 |
| CHEMBL1444820 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1364011 | — | EC50 | = | 106.0 | nM | 6.97 |
| CHEMBL1537542 | — | EC50 | = | 106.0 | nM | 6.97 |
| CHEMBL1485275 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL1422253 | — | EC50 | = | 111.0 | nM | 6.96 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL1382674 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL1237072 | DIRITHROMYCIN | EC50 | = | 117.0 | nM | 6.93 |
| CHEMBL1318922 | — | EC50 | = | 117.0 | nM | 6.93 |
| CHEMBL1484438 | — | EC50 | = | 124.0 | nM | 6.91 |
| CHEMBL1516396 | — | EC50 | = | 125.0 | nM | 6.90 |
| CHEMBL1256686 | CALCIMYCIN | EC50 | = | 128.0 | nM | 6.89 |
| CHEMBL287542 | RAFOXANIDE | EC50 | = | 137.0 | nM | 6.86 |
| CHEMBL1528206 | — | EC50 | = | 141.0 | nM | 6.85 |
| CHEMBL278255 | CLINAFLOXACIN | EC50 | = | 142.0 | nM | 6.85 |
| CHEMBL2146063 | CHLORTETRACYCLINE HYDROCHLORIDE | EC50 | = | 148.0 | nM | 6.83 |
| CHEMBL1344339 | — | EC50 | = | 147.0 | nM | 6.83 |
| CHEMBL1342436 | — | EC50 | = | 153.0 | nM | 6.82 |
| CHEMBL1583292 | — | EC50 | = | 167.0 | nM | 6.78 |
| CHEMBL1385808 | — | EC50 | = | 173.0 | nM | 6.76 |
| CHEMBL1545940 | — | EC50 | = | 184.0 | nM | 6.74 |
| CHEMBL1333965 | — | EC50 | = | 182.0 | nM | 6.74 |
| CHEMBL1326397 | — | EC50 | = | 228.0 | nM | 6.64 |
| CHEMBL1493936 | — | EC50 | = | 228.0 | nM | 6.64 |
| CHEMBL1576581 | — | EC50 | = | 229.0 | nM | 6.64 |
| CHEMBL1319643 | — | EC50 | = | 245.0 | nM | 6.61 |
| CHEMBL1417731 | — | EC50 | = | 257.0 | nM | 6.59 |
| CHEMBL589238 | — | EC50 | = | 254.0 | nM | 6.59 |
| CHEMBL1452449 | — | EC50 | = | 264.0 | nM | 6.58 |
| CHEMBL496 | HEXACHLOROPHENE | EC50 | = | 262.0 | nM | 6.58 |
| CHEMBL1509369 | — | EC50 | = | 269.0 | nM | 6.57 |
| CHEMBL1551640 | — | EC50 | = | 277.0 | nM | 6.56 |
| CHEMBL1545189 | — | EC50 | = | 283.0 | nM | 6.55 |
| CHEMBL1572266 | — | EC50 | = | 299.0 | nM | 6.52 |
| CHEMBL1431875 | — | EC50 | = | 316.0 | nM | 6.50 |
| CHEMBL1373646 | — | EC50 | = | 337.0 | nM | 6.47 |
| CHEMBL1521292 | — | EC50 | = | 341.0 | nM | 6.47 |
| CHEMBL3198213 | — | EC50 | = | 350.0 | nM | 6.46 |
| CHEMBL1542263 | — | EC50 | = | 343.0 | nM | 6.46 |
| CHEMBL1299389 | — | EC50 | = | 344.0 | nM | 6.46 |
| CHEMBL1200735 | MOXIFLOXACIN HYDROCHLORIDE | EC50 | = | 358.0 | nM | 6.45 |
| CHEMBL1570738 | — | EC50 | = | 372.0 | nM | 6.43 |
| CHEMBL1314141 | — | EC50 | = | 384.0 | nM | 6.42 |
| CHEMBL1482975 | — | EC50 | = | 421.0 | nM | 6.38 |