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Compound Detail

CHEMBL1542263

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CC(C(=O)NC1C(=O)N2C(C(=O)O)=C(CSc3nnnn3C)CSC12)n1cc(Cl)cn1

Basic Information

ChEMBL ID CHEMBL1542263
Phase Preclinical
Structure Type MOL
InChI Key SRFXZBVHYQPYLN-UHFFFAOYSA-N
3
Targets
3
Activities
1
Assay Types
0
PK Parameters
0
Publications
0
Known Names

Molecular Properties

484.9
MW (Da)
0.15
ALogP
11
HBA
2
HBD
148.1
PSA (Ų)
0.41
QED
1
Ro5 Violations
7
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

First in Class Prodrug

Extended Properties

Molecular Formula C16H17ClN8O4S2
MW 484.95
Aromatic Rings 2
Heavy Atoms 31
NP-Likeness -1.65

Activity Summary

EC50 3 meas. best 7.11

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Streptokinase A
CHEMBL1293228
EC50 7.11 7.11 78.0 1
Streptococcus sp. 'group A'
CHEMBL612389
EC50 6.79 6.79 161.0 1
Streptococcus
CHEMBL612313
EC50 6.46 6.46 343.0 1

Activity Data Samples

Top measurements by pChEMBL value

Data from ChEMBL 36 via Core Engine