Assay Detail
Functional
CHEMBL1614064
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Confirmation HTS to Identify Inhibitors of Streptokinase Promotor Activity. (Class of assay: confirmatory) [Related pubchem assays: 1677 (Project Summary), 1662 (Primary HTS)]
3226
Total Activities
3223
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Streptococcus pyogenes M1 GAS |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Streptokinase A (CHEMBL1293228) ↗| Type | SINGLE PROTEIN |
| Organism | Streptococcus pyogenes serotype M1 |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3226 | 5.48 | 7.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2094567 | — | — | 1 | 7.20 |
| CHEMBL2146063 | CHLORTETRACYCLINE HYDROCHLORIDE | 4.0 | 1 | 7.19 |
| CHEMBL278255 | CLINAFLOXACIN | 2.0 | 1 | 7.19 |
| CHEMBL1422078 | — | — | 1 | 7.16 |
| CHEMBL1427178 | — | — | 1 | 7.13 |
| CHEMBL1593888 | — | — | 1 | 7.13 |
| CHEMBL1542263 | — | — | 1 | 7.11 |
| CHEMBL12131 | CLOSANTEL | 2.0 | 1 | 7.09 |
| CHEMBL1306986 | — | — | 1 | 7.09 |
| CHEMBL1563791 | — | — | 1 | 7.05 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | 4.0 | 1 | 7.03 |
| CHEMBL1385808 | — | — | 1 | 7.02 |
| CHEMBL1334646 | — | — | 1 | 7.02 |
| CHEMBL3197065 | — | — | 1 | 7.02 |
| CHEMBL1545940 | — | — | 1 | 7.02 |
| CHEMBL1551640 | — | — | 1 | 7.02 |
| CHEMBL1349631 | — | — | 1 | 7.01 |
| CHEMBL1319643 | — | — | 1 | 7.01 |
| CHEMBL1578607 | — | — | 1 | 7.01 |
| CHEMBL1381242 | — | — | 1 | 7.00 |
| CHEMBL1539595 | — | — | 1 | 6.99 |
| CHEMBL1522288 | — | — | 1 | 6.98 |
| CHEMBL1583292 | — | — | 1 | 6.97 |
| CHEMBL583584 | — | — | 1 | 6.96 |
| CHEMBL1458477 | — | — | 1 | 6.96 |
| CHEMBL1299389 | — | — | 1 | 6.95 |
| CHEMBL1562033 | — | — | 1 | 6.94 |
| CHEMBL1484438 | — | — | 1 | 6.94 |
| CHEMBL1407169 | — | — | 1 | 6.94 |
| CHEMBL1525098 | — | — | 1 | 6.94 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2094567 | — | EC50 | = | 63.0 | nM | 7.20 |
| CHEMBL2146063 | CHLORTETRACYCLINE HYDROCHLORIDE | EC50 | = | 65.0 | nM | 7.19 |
| CHEMBL278255 | CLINAFLOXACIN | EC50 | = | 64.0 | nM | 7.19 |
| CHEMBL1422078 | — | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL1593888 | — | EC50 | = | 74.0 | nM | 7.13 |
| CHEMBL1427178 | — | EC50 | = | 74.0 | nM | 7.13 |
| CHEMBL1542263 | — | EC50 | = | 78.0 | nM | 7.11 |
| CHEMBL1306986 | — | EC50 | = | 81.0 | nM | 7.09 |
| CHEMBL12131 | CLOSANTEL | EC50 | = | 82.0 | nM | 7.09 |
| CHEMBL1563791 | — | EC50 | = | 90.0 | nM | 7.05 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | EC50 | = | 93.0 | nM | 7.03 |
| CHEMBL3197065 | — | EC50 | = | 95.0 | nM | 7.02 |
| CHEMBL1334646 | — | EC50 | = | 96.0 | nM | 7.02 |
| CHEMBL1545940 | — | EC50 | = | 96.0 | nM | 7.02 |
| CHEMBL1385808 | — | EC50 | = | 95.0 | nM | 7.02 |
| CHEMBL1551640 | — | EC50 | = | 95.0 | nM | 7.02 |
| CHEMBL1319643 | — | EC50 | = | 98.0 | nM | 7.01 |
| CHEMBL1578607 | — | EC50 | = | 97.0 | nM | 7.01 |
| CHEMBL1349631 | — | EC50 | = | 98.0 | nM | 7.01 |
| CHEMBL1381242 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1539595 | — | EC50 | = | 102.0 | nM | 6.99 |
| CHEMBL1522288 | — | EC50 | = | 105.0 | nM | 6.98 |
| CHEMBL1583292 | — | EC50 | = | 108.0 | nM | 6.97 |
| CHEMBL583584 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL1458477 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL1299389 | — | EC50 | = | 112.0 | nM | 6.95 |
| CHEMBL1484438 | — | EC50 | = | 114.0 | nM | 6.94 |
| CHEMBL1407169 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL1525098 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL1562033 | — | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL1314141 | — | EC50 | = | 119.0 | nM | 6.92 |
| CHEMBL1436772 | — | EC50 | = | 127.0 | nM | 6.90 |
| CHEMBL127 | MEROPENEM | EC50 | = | 127.0 | nM | 6.90 |
| CHEMBL1344339 | — | EC50 | = | 127.0 | nM | 6.90 |
| CHEMBL1570738 | — | EC50 | = | 128.0 | nM | 6.89 |
| CHEMBL1509369 | — | EC50 | = | 130.0 | nM | 6.89 |
| CHEMBL1324005 | — | EC50 | = | 131.0 | nM | 6.88 |
| CHEMBL1366997 | — | EC50 | = | 134.0 | nM | 6.87 |
| CHEMBL1390121 | — | EC50 | = | 136.0 | nM | 6.87 |
| CHEMBL1334568 | — | EC50 | = | 139.0 | nM | 6.86 |
| CHEMBL1304666 | — | EC50 | = | 138.0 | nM | 6.86 |
| CHEMBL1455627 | — | EC50 | = | 137.0 | nM | 6.86 |
| CHEMBL1482975 | — | EC50 | = | 140.0 | nM | 6.85 |
| CHEMBL1405262 | — | EC50 | = | 142.0 | nM | 6.85 |
| CHEMBL1412157 | — | EC50 | = | 145.0 | nM | 6.84 |
| CHEMBL1452449 | — | EC50 | = | 144.0 | nM | 6.84 |
| CHEMBL1546739 | — | EC50 | = | 145.0 | nM | 6.84 |
| CHEMBL1595820 | — | EC50 | = | 149.0 | nM | 6.83 |
| CHEMBL1200596 | CHLOROXINE | EC50 | = | 148.0 | nM | 6.83 |
| CHEMBL1456111 | — | EC50 | = | 149.0 | nM | 6.83 |