Assay Detail
Functional
CHEMBL1613983
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Microorganism-Based Dose Confirmation HTS to Identify Compounds Cytotoxic to SK(-)GAS Group A Streptococcus. (Class of assay: confirmatory) [Related pubchem assays: 1677 (Project Summary), 1662 (Primary HTS)]
3222
Total Activities
3219
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Streptococcus |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Target
Streptococcus sp. 'group A' (CHEMBL612389) ↗| Type | ORGANISM |
| Organism | Streptococcus sp. 'group A' |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3222 | 5.40 | 7.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1452261 | — | — | 1 | 7.20 |
| CHEMBL1463750 | — | — | 1 | 7.17 |
| CHEMBL1350780 | — | — | 1 | 7.17 |
| CHEMBL1376248 | — | — | 1 | 7.16 |
| CHEMBL1517362 | — | — | 1 | 7.14 |
| CHEMBL1431875 | — | — | 1 | 7.14 |
| CHEMBL1456111 | — | — | 1 | 7.13 |
| CHEMBL1525098 | — | — | 1 | 7.13 |
| CHEMBL1545940 | — | — | 1 | 7.11 |
| CHEMBL287542 | RAFOXANIDE | 2.0 | 1 | 7.10 |
| CHEMBL1385808 | — | — | 1 | 7.10 |
| CHEMBL1551640 | — | — | 1 | 7.06 |
| CHEMBL1537542 | — | — | 1 | 7.05 |
| CHEMBL1578607 | — | — | 1 | 7.00 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | 4.0 | 1 | 7.00 |
| CHEMBL1545189 | — | — | 1 | 7.00 |
| CHEMBL2094567 | — | — | 1 | 7.00 |
| CHEMBL1334646 | — | — | 1 | 7.00 |
| CHEMBL1516396 | — | — | 1 | 7.00 |
| CHEMBL589238 | — | — | 1 | 6.98 |
| CHEMBL1319643 | — | — | 1 | 6.96 |
| CHEMBL3195767 | — | — | 1 | 6.96 |
| CHEMBL1484438 | — | — | 1 | 6.96 |
| CHEMBL1373646 | — | — | 1 | 6.95 |
| CHEMBL12131 | CLOSANTEL | 2.0 | 1 | 6.94 |
| CHEMBL278255 | CLINAFLOXACIN | 2.0 | 1 | 6.94 |
| CHEMBL1609946 | — | — | 1 | 6.92 |
| CHEMBL1366997 | — | — | 1 | 6.91 |
| CHEMBL1458477 | — | — | 1 | 6.90 |
| CHEMBL1411241 | — | — | 1 | 6.86 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1452261 | — | EC50 | = | 63.0 | nM | 7.20 |
| CHEMBL1350780 | — | EC50 | = | 68.0 | nM | 7.17 |
| CHEMBL1463750 | — | EC50 | = | 67.0 | nM | 7.17 |
| CHEMBL1376248 | — | EC50 | = | 69.0 | nM | 7.16 |
| CHEMBL1517362 | — | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL1431875 | — | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL1456111 | — | EC50 | = | 74.0 | nM | 7.13 |
| CHEMBL1525098 | — | EC50 | = | 74.0 | nM | 7.13 |
| CHEMBL1545940 | — | EC50 | = | 78.0 | nM | 7.11 |
| CHEMBL1385808 | — | EC50 | = | 79.0 | nM | 7.10 |
| CHEMBL287542 | RAFOXANIDE | EC50 | = | 80.0 | nM | 7.10 |
| CHEMBL1551640 | — | EC50 | = | 88.0 | nM | 7.06 |
| CHEMBL1537542 | — | EC50 | = | 90.0 | nM | 7.05 |
| CHEMBL1516396 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1545189 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL1578607 | — | EC50 | = | 99.0 | nM | 7.00 |
| CHEMBL1334646 | — | EC50 | = | 99.0 | nM | 7.00 |
| CHEMBL2094567 | — | EC50 | = | 99.0 | nM | 7.00 |
| CHEMBL2146123 | METHACYCLINE HYDROCHLORIDE | EC50 | = | 99.0 | nM | 7.00 |
| CHEMBL589238 | — | EC50 | = | 104.0 | nM | 6.98 |
| CHEMBL1484438 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL1319643 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL3195767 | — | EC50 | = | 109.0 | nM | 6.96 |
| CHEMBL1373646 | — | EC50 | = | 112.0 | nM | 6.95 |
| CHEMBL278255 | CLINAFLOXACIN | EC50 | = | 115.0 | nM | 6.94 |
| CHEMBL12131 | CLOSANTEL | EC50 | = | 114.0 | nM | 6.94 |
| CHEMBL1609946 | — | EC50 | = | 120.0 | nM | 6.92 |
| CHEMBL1366997 | — | EC50 | = | 124.0 | nM | 6.91 |
| CHEMBL1458477 | — | EC50 | = | 127.0 | nM | 6.90 |
| CHEMBL1411241 | — | EC50 | = | 138.0 | nM | 6.86 |
| CHEMBL1483146 | — | EC50 | = | 137.0 | nM | 6.86 |
| CHEMBL1407169 | — | EC50 | = | 148.0 | nM | 6.83 |
| CHEMBL127 | MEROPENEM | EC50 | = | 153.0 | nM | 6.82 |
| CHEMBL1470448 | — | EC50 | = | 159.0 | nM | 6.80 |
| CHEMBL1542263 | — | EC50 | = | 161.0 | nM | 6.79 |
| CHEMBL1334456 | — | EC50 | = | 161.0 | nM | 6.79 |
| CHEMBL1349631 | — | EC50 | = | 165.0 | nM | 6.78 |
| CHEMBL1509369 | — | EC50 | = | 169.0 | nM | 6.77 |
| CHEMBL126 | LINEZOLID | EC50 | = | 170.0 | nM | 6.77 |
| CHEMBL1314141 | — | EC50 | = | 175.0 | nM | 6.76 |
| CHEMBL1324005 | — | EC50 | = | 179.0 | nM | 6.75 |
| CHEMBL1576581 | — | EC50 | = | 179.0 | nM | 6.75 |
| CHEMBL1522288 | — | EC50 | = | 181.0 | nM | 6.74 |
| CHEMBL1427178 | — | EC50 | = | 182.0 | nM | 6.74 |
| CHEMBL1595820 | — | EC50 | = | 186.0 | nM | 6.73 |
| CHEMBL590947 | — | EC50 | = | 192.0 | nM | 6.72 |
| CHEMBL1447284 | — | EC50 | = | 191.0 | nM | 6.72 |
| CHEMBL1519902 | — | EC50 | = | 190.0 | nM | 6.72 |
| CHEMBL1572510 | — | EC50 | = | 195.0 | nM | 6.71 |
| CHEMBL1563791 | — | EC50 | = | 196.0 | nM | 6.71 |