Assay Detail
Binding
CHEMBL1738418
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence-based biochemical high throughput dose response assay for activators of the calcium sensitivity of cardiac Regulated Thin Filaments (RTF). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493008, AID493018, AID504382, AID504383]
244
Total Activities
244
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 244 | 5.42 | 6.78 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1581326 | — | — | 1 | 6.78 |
| CHEMBL3195681 | — | — | 1 | 6.78 |
| CHEMBL3195851 | — | — | 1 | 6.72 |
| CHEMBL1468444 | — | — | 1 | 6.55 |
| CHEMBL1379673 | — | — | 1 | 6.54 |
| CHEMBL1477915 | — | — | 1 | 6.40 |
| CHEMBL1398812 | — | — | 1 | 6.38 |
| CHEMBL1369691 | — | — | 1 | 6.30 |
| CHEMBL1573529 | — | — | 1 | 6.29 |
| CHEMBL3197404 | — | — | 1 | 6.25 |
| CHEMBL1388372 | — | — | 1 | 6.21 |
| CHEMBL1604510 | — | — | 1 | 6.13 |
| CHEMBL1550816 | — | — | 1 | 6.12 |
| CHEMBL1725987 | — | — | 1 | 6.07 |
| CHEMBL1586687 | — | — | 1 | 6.06 |
| CHEMBL1975147 | — | — | 1 | 5.96 |
| CHEMBL1313968 | — | — | 1 | 5.95 |
| CHEMBL1429070 | — | — | 1 | 5.94 |
| CHEMBL1310204 | — | — | 1 | 5.94 |
| CHEMBL1713654 | — | — | 1 | 5.92 |
| CHEMBL1501273 | — | — | 1 | 5.86 |
| CHEMBL1977499 | — | — | 1 | 5.84 |
| CHEMBL1499258 | — | — | 1 | 5.83 |
| CHEMBL1542169 | — | — | 1 | 5.81 |
| CHEMBL1574521 | — | — | 1 | 5.81 |
| CHEMBL1407632 | — | — | 1 | 5.80 |
| CHEMBL1586067 | — | — | 1 | 5.74 |
| CHEMBL1971695 | — | — | 1 | 5.73 |
| CHEMBL1576905 | — | — | 1 | 5.73 |
| CHEMBL1701437 | — | — | 1 | 5.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1581326 | — | EC50 | = | 165.07 | nM | 6.78 |
| CHEMBL3195681 | — | EC50 | = | 164.57 | nM | 6.78 |
| CHEMBL3195851 | — | EC50 | = | 190.67 | nM | 6.72 |
| CHEMBL1468444 | — | EC50 | = | 278.85 | nM | 6.55 |
| CHEMBL1379673 | — | EC50 | = | 286.87 | nM | 6.54 |
| CHEMBL1477915 | — | EC50 | = | 396.99 | nM | 6.40 |
| CHEMBL1398812 | — | EC50 | = | 413.02 | nM | 6.38 |
| CHEMBL1369691 | — | EC50 | = | 500.48 | nM | 6.30 |
| CHEMBL1573529 | — | EC50 | = | 515.79 | nM | 6.29 |
| CHEMBL3197404 | — | EC50 | = | 565.38 | nM | 6.25 |
| CHEMBL1388372 | — | EC50 | = | 615.36 | nM | 6.21 |
| CHEMBL1604510 | — | EC50 | = | 742.02 | nM | 6.13 |
| CHEMBL1550816 | — | EC50 | = | 760.72 | nM | 6.12 |
| CHEMBL1725987 | — | EC50 | = | 852.88 | nM | 6.07 |
| CHEMBL1586687 | — | EC50 | = | 869.62 | nM | 6.06 |
| CHEMBL1975147 | — | EC50 | = | 1101.0 | nM | 5.96 |
| CHEMBL1313968 | — | EC50 | = | 1113.0 | nM | 5.95 |
| CHEMBL1429070 | — | EC50 | = | 1143.0 | nM | 5.94 |
| CHEMBL1310204 | — | EC50 | = | 1137.0 | nM | 5.94 |
| CHEMBL1713654 | — | EC50 | = | 1209.0 | nM | 5.92 |
| CHEMBL1501273 | — | EC50 | = | 1369.0 | nM | 5.86 |
| CHEMBL1977499 | — | EC50 | = | 1438.0 | nM | 5.84 |
| CHEMBL1499258 | — | EC50 | = | 1465.0 | nM | 5.83 |
| CHEMBL1574521 | — | EC50 | = | 1548.0 | nM | 5.81 |
| CHEMBL1542169 | — | EC50 | = | 1537.0 | nM | 5.81 |
| CHEMBL1407632 | — | EC50 | = | 1577.0 | nM | 5.80 |
| CHEMBL1586067 | — | EC50 | = | 1830.0 | nM | 5.74 |
| CHEMBL1576905 | — | EC50 | = | 1878.0 | nM | 5.73 |
| CHEMBL1971695 | — | EC50 | = | 1863.0 | nM | 5.73 |
| CHEMBL1701437 | — | EC50 | = | 1981.0 | nM | 5.70 |
| CHEMBL1466913 | — | EC50 | = | 2022.0 | nM | 5.69 |
| CHEMBL1576602 | — | EC50 | = | 2177.0 | nM | 5.66 |
| CHEMBL1462008 | — | EC50 | = | 2218.0 | nM | 5.65 |
| CHEMBL1540557 | — | EC50 | = | 2385.0 | nM | 5.62 |
| CHEMBL1466606 | — | EC50 | = | 2576.0 | nM | 5.59 |
| CHEMBL1725983 | — | EC50 | = | 2574.0 | nM | 5.59 |
| CHEMBL1557186 | — | EC50 | = | 2706.0 | nM | 5.57 |
| CHEMBL2004884 | — | EC50 | = | 2780.0 | nM | 5.56 |
| CHEMBL1547468 | — | EC50 | = | 2901.0 | nM | 5.54 |
| CHEMBL1311198 | — | EC50 | = | 2918.0 | nM | 5.54 |
| CHEMBL1596655 | — | EC50 | = | 3326.0 | nM | 5.48 |
| CHEMBL2001481 | — | EC50 | = | 3708.0 | nM | 5.43 |
| CHEMBL1594911 | — | EC50 | = | 3734.0 | nM | 5.43 |
| CHEMBL1970784 | — | EC50 | = | 3934.0 | nM | 5.41 |
| CHEMBL2002008 | — | EC50 | = | 3911.0 | nM | 5.41 |
| CHEMBL1342181 | — | EC50 | = | 4162.0 | nM | 5.38 |
| CHEMBL1991136 | — | EC50 | = | 4497.0 | nM | 5.35 |
| CHEMBL1580769 | — | EC50 | = | 4529.0 | nM | 5.34 |
| CHEMBL1504676 | — | EC50 | = | 4888.0 | nM | 5.31 |
| CHEMBL1316798 | — | EC50 | = | 4962.0 | nM | 5.30 |