Assay Detail
Functional
CHEMBL1738423
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR analysis of Ubc13-Ubiquitination selectivity in a TR-FRET assay for In Vitro dose response studies. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2006, AID2011, AID2018, AID2069, AID2614]
114
Total Activities
110
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 114 | 4.26 | 4.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL273264 | NAFAMOSTAT | 3.0 | 1 | 4.85 |
| CHEMBL1706280 | — | — | 2 | 4.78 |
| CHEMBL1706577 | — | — | 2 | 4.63 |
| CHEMBL1704267 | — | — | 2 | 4.58 |
| CHEMBL1699571 | — | — | 1 | 4.48 |
| CHEMBL1308068 | — | — | 1 | 4.46 |
| CHEMBL1399979 | — | — | 1 | 4.33 |
| CHEMBL1402286 | — | — | 1 | 4.27 |
| CHEMBL1546410 | — | — | 1 | 4.27 |
| CHEMBL1728000 | — | — | 1 | 4.23 |
| CHEMBL1361703 | — | — | 1 | 4.22 |
| CHEMBL1700951 | — | — | 1 | 4.19 |
| CHEMBL1725449 | — | — | 1 | 4.17 |
| CHEMBL1720079 | — | — | 1 | 4.14 |
| CHEMBL1736986 | — | — | 1 | 4.14 |
| CHEMBL1731605 | — | — | 2 | 4.13 |
| CHEMBL1562713 | — | — | 1 | 4.11 |
| CHEMBL1722076 | — | — | 1 | 4.09 |
| CHEMBL1731180 | — | — | 1 | 4.08 |
| CHEMBL1706851 | — | — | 1 | 4.08 |
| CHEMBL1727666 | — | — | 1 | 4.07 |
| CHEMBL1706750 | — | — | 1 | 4.06 |
| CHEMBL1719957 | — | — | 1 | 4.03 |
| CHEMBL1518374 | — | — | 1 | 4.03 |
| CHEMBL1735822 | — | — | 1 | 4.03 |
| CHEMBL1374955 | — | — | 1 | 4.01 |
| CHEMBL1372651 | — | — | 1 | 4.01 |
| CHEMBL1707853 | — | — | 1 | - |
| CHEMBL1417070 | — | — | 1 | - |
| CHEMBL1368287 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL273264 | NAFAMOSTAT | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL1706280 | — | IC50 | = | 16700.0 | nM | 4.78 |
| CHEMBL1706577 | — | IC50 | = | 23300.0 | nM | 4.63 |
| CHEMBL1706577 | — | IC50 | = | 25800.0 | nM | 4.59 |
| CHEMBL1704267 | — | IC50 | = | 26100.0 | nM | 4.58 |
| CHEMBL1704267 | — | IC50 | = | 31200.0 | nM | 4.51 |
| CHEMBL1699571 | — | IC50 | = | 33100.0 | nM | 4.48 |
| CHEMBL1308068 | — | IC50 | = | 34600.0 | nM | 4.46 |
| CHEMBL1399979 | — | IC50 | = | 47200.0 | nM | 4.33 |
| CHEMBL1402286 | — | IC50 | = | 53400.0 | nM | 4.27 |
| CHEMBL1546410 | — | IC50 | = | 53800.0 | nM | 4.27 |
| CHEMBL1728000 | — | IC50 | = | 58900.0 | nM | 4.23 |
| CHEMBL1361703 | — | IC50 | = | 60200.0 | nM | 4.22 |
| CHEMBL1700951 | — | IC50 | = | 65000.0 | nM | 4.19 |
| CHEMBL1725449 | — | IC50 | = | 68200.0 | nM | 4.17 |
| CHEMBL1736986 | — | IC50 | = | 72500.0 | nM | 4.14 |
| CHEMBL1720079 | — | IC50 | = | 72700.0 | nM | 4.14 |
| CHEMBL1731605 | — | IC50 | = | 74400.0 | nM | 4.13 |
| CHEMBL1731605 | — | IC50 | = | 73400.0 | nM | 4.13 |
| CHEMBL1562713 | — | IC50 | = | 78400.0 | nM | 4.11 |
| CHEMBL1722076 | — | IC50 | = | 81100.0 | nM | 4.09 |
| CHEMBL1706851 | — | IC50 | = | 83000.0 | nM | 4.08 |
| CHEMBL1731180 | — | IC50 | = | 82500.0 | nM | 4.08 |
| CHEMBL1727666 | — | IC50 | = | 86100.0 | nM | 4.07 |
| CHEMBL1706750 | — | IC50 | = | 86600.0 | nM | 4.06 |
| CHEMBL1518374 | — | IC50 | = | 93100.0 | nM | 4.03 |
| CHEMBL1719957 | — | IC50 | = | 92600.0 | nM | 4.03 |
| CHEMBL1735822 | — | IC50 | = | 92600.0 | nM | 4.03 |
| CHEMBL1372651 | — | IC50 | = | 98500.0 | nM | 4.01 |
| CHEMBL1374955 | — | IC50 | = | 98000.0 | nM | 4.01 |
| CHEMBL1727199 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1446655 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1381243 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1716258 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1342081 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL390401 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1418005 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1714309 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1519689 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1378427 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1448519 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1733948 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1713480 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1733142 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1703530 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1722739 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1464539 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1405964 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1736753 | — | IC50 | > | 100000.0 | nM | - |
| CHEMBL1703238 | — | IC50 | > | 100000.0 | nM | - |