Assay Detail
Functional
CHEMBL1738428
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR analysis of inhibitors of TNFa specific NF-kB induction - Set 3. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1575, AID1578, AID1852, AID2335, AID2337, AID2483]
40
Total Activities
39
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 40 | 5.02 | 5.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1331314 | — | — | 1 | 5.67 |
| CHEMBL1444568 | — | — | 1 | 5.47 |
| CHEMBL1452157 | — | — | 1 | 5.25 |
| CHEMBL1346587 | — | — | 1 | 4.99 |
| CHEMBL1336829 | — | — | 1 | 4.89 |
| CHEMBL1732655 | — | — | 1 | 4.75 |
| CHEMBL1519375 | — | — | 2 | 4.74 |
| CHEMBL1700774 | — | — | 1 | 4.70 |
| CHEMBL1305184 | — | — | 1 | - |
| CHEMBL1699939 | — | — | 1 | - |
| CHEMBL1363341 | — | — | 1 | - |
| CHEMBL1412853 | — | — | 1 | - |
| CHEMBL1700576 | — | — | 1 | - |
| CHEMBL1698072 | — | — | 1 | - |
| CHEMBL1299367 | — | — | 1 | - |
| CHEMBL1345225 | — | — | 1 | - |
| CHEMBL1515929 | — | — | 1 | - |
| CHEMBL1719080 | — | — | 1 | - |
| CHEMBL1468879 | — | — | 1 | - |
| CHEMBL1733730 | — | — | 1 | - |
| CHEMBL1448844 | — | — | 1 | - |
| CHEMBL1726554 | — | — | 1 | - |
| CHEMBL1386167 | — | — | 1 | - |
| CHEMBL1705192 | — | — | 1 | - |
| CHEMBL1491481 | — | — | 1 | - |
| CHEMBL1354593 | — | — | 1 | - |
| CHEMBL1711872 | — | — | 1 | - |
| CHEMBL1725059 | — | — | 1 | - |
| CHEMBL1394462 | — | — | 1 | - |
| CHEMBL1725440 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1331314 | — | IC50 | = | 2120.0 | nM | 5.67 |
| CHEMBL1444568 | — | IC50 | = | 3350.0 | nM | 5.47 |
| CHEMBL1452157 | — | IC50 | = | 5660.0 | nM | 5.25 |
| CHEMBL1346587 | — | IC50 | = | 10300.0 | nM | 4.99 |
| CHEMBL1336829 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL1732655 | — | IC50 | = | 17700.0 | nM | 4.75 |
| CHEMBL1519375 | — | IC50 | = | 18200.0 | nM | 4.74 |
| CHEMBL1519375 | — | IC50 | = | 18600.0 | nM | 4.73 |
| CHEMBL1700774 | — | IC50 | = | 19900.0 | nM | 4.70 |
| CHEMBL1299367 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1711872 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1345225 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1515929 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1719080 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1468879 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1699939 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1314651 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1702956 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1327036 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1567543 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1595049 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1711631 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1731457 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1397246 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1698072 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1700576 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1412853 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1363341 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1305184 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1733730 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1448844 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1386167 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1726554 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1705192 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1491481 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1354593 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1725059 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1702238 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1394462 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1725440 | — | IC50 | > | 20000.0 | nM | - |