Assay Detail
Functional
CHEMBL1738430
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of Image-Based HTS for Selective Agonists for NTR1. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493036, AID493055]
185
Total Activities
185
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 185 | 4.89 | 5.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1501508 | — | — | 1 | 5.62 |
| CHEMBL1442136 | — | — | 1 | 5.60 |
| CHEMBL1601394 | — | — | 1 | 5.57 |
| CHEMBL1577981 | — | — | 1 | 5.54 |
| CHEMBL1301125 | — | — | 1 | 5.49 |
| CHEMBL1323442 | — | — | 1 | 5.47 |
| CHEMBL1308657 | — | — | 1 | 5.45 |
| CHEMBL1490404 | — | — | 1 | 5.42 |
| CHEMBL1611170 | — | — | 1 | 5.41 |
| CHEMBL1600146 | — | — | 1 | 5.41 |
| CHEMBL1468368 | — | — | 1 | 5.38 |
| CHEMBL1540679 | — | — | 1 | 5.38 |
| CHEMBL1299997 | — | — | 1 | 5.37 |
| CHEMBL508338 | THIMEROSAL | 3.0 | 1 | 5.36 |
| CHEMBL1546134 | — | — | 1 | 5.29 |
| CHEMBL532160 | — | — | 1 | 5.27 |
| CHEMBL1538066 | — | — | 1 | 5.27 |
| CHEMBL1303193 | — | — | 1 | 5.24 |
| CHEMBL1589062 | — | — | 1 | 5.24 |
| CHEMBL1597454 | — | — | 1 | 5.23 |
| CHEMBL1547420 | — | — | 1 | 5.22 |
| CHEMBL1312502 | — | — | 1 | 5.22 |
| CHEMBL1586252 | — | — | 1 | 5.21 |
| CHEMBL1446377 | — | — | 1 | 5.21 |
| CHEMBL1328169 | — | — | 1 | 5.21 |
| CHEMBL1594369 | — | — | 1 | 5.18 |
| CHEMBL1613675 | — | — | 1 | 5.18 |
| CHEMBL3210863 | — | — | 1 | 5.18 |
| CHEMBL2003819 | — | — | 1 | 5.18 |
| CHEMBL1550591 | — | — | 1 | 5.18 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1501508 | — | EC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL1442136 | — | EC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL1601394 | — | EC50 | = | 2710.0 | nM | 5.57 |
| CHEMBL1577981 | — | EC50 | = | 2910.0 | nM | 5.54 |
| CHEMBL1301125 | — | EC50 | = | 3270.0 | nM | 5.49 |
| CHEMBL1323442 | — | EC50 | = | 3350.0 | nM | 5.47 |
| CHEMBL1308657 | — | EC50 | = | 3590.0 | nM | 5.45 |
| CHEMBL1490404 | — | EC50 | = | 3800.0 | nM | 5.42 |
| CHEMBL1600146 | — | EC50 | = | 3910.0 | nM | 5.41 |
| CHEMBL1611170 | — | EC50 | = | 3890.0 | nM | 5.41 |
| CHEMBL1468368 | — | EC50 | = | 4120.0 | nM | 5.38 |
| CHEMBL1540679 | — | EC50 | = | 4160.0 | nM | 5.38 |
| CHEMBL1299997 | — | EC50 | = | 4260.0 | nM | 5.37 |
| CHEMBL508338 | THIMEROSAL | EC50 | = | 4370.0 | nM | 5.36 |
| CHEMBL1546134 | — | EC50 | = | 5140.0 | nM | 5.29 |
| CHEMBL1538066 | — | EC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL532160 | — | EC50 | = | 5350.0 | nM | 5.27 |
| CHEMBL1589062 | — | EC50 | = | 5720.0 | nM | 5.24 |
| CHEMBL1303193 | — | EC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL1597454 | — | EC50 | = | 5830.0 | nM | 5.23 |
| CHEMBL1547420 | — | EC50 | = | 5980.0 | nM | 5.22 |
| CHEMBL1312502 | — | EC50 | = | 6000.0 | nM | 5.22 |
| CHEMBL1328169 | — | EC50 | = | 6210.0 | nM | 5.21 |
| CHEMBL1446377 | — | EC50 | = | 6190.0 | nM | 5.21 |
| CHEMBL1586252 | — | EC50 | = | 6240.0 | nM | 5.21 |
| CHEMBL3210863 | — | EC50 | = | 6650.0 | nM | 5.18 |
| CHEMBL1613675 | — | EC50 | = | 6650.0 | nM | 5.18 |
| CHEMBL1550591 | — | EC50 | = | 6660.0 | nM | 5.18 |
| CHEMBL1594369 | — | EC50 | = | 6590.0 | nM | 5.18 |
| CHEMBL2003819 | — | EC50 | = | 6620.0 | nM | 5.18 |
| CHEMBL1483562 | — | EC50 | = | 6690.0 | nM | 5.17 |
| CHEMBL1966869 | — | EC50 | = | 7150.0 | nM | 5.15 |
| CHEMBL1611686 | — | EC50 | = | 7490.0 | nM | 5.13 |
| CHEMBL1438069 | — | EC50 | = | 7370.0 | nM | 5.13 |
| CHEMBL1595121 | — | EC50 | = | 7500.0 | nM | 5.12 |
| CHEMBL1340713 | — | EC50 | = | 7590.0 | nM | 5.12 |
| CHEMBL1453900 | — | EC50 | = | 7590.0 | nM | 5.12 |
| CHEMBL1461496 | — | EC50 | = | 7860.0 | nM | 5.11 |
| CHEMBL1387563 | — | EC50 | = | 7890.0 | nM | 5.10 |
| CHEMBL1385214 | — | EC50 | = | 8210.0 | nM | 5.09 |
| CHEMBL1321527 | — | EC50 | = | 8090.0 | nM | 5.09 |
| CHEMBL1369296 | — | EC50 | = | 8290.0 | nM | 5.08 |
| CHEMBL1995726 | — | EC50 | = | 8510.0 | nM | 5.07 |
| CHEMBL1550862 | — | EC50 | = | 8480.0 | nM | 5.07 |
| CHEMBL1502512 | — | EC50 | = | 8730.0 | nM | 5.06 |
| CHEMBL1608453 | — | EC50 | = | 8640.0 | nM | 5.06 |
| CHEMBL1586169 | — | EC50 | = | 8850.0 | nM | 5.05 |
| CHEMBL1493442 | — | EC50 | = | 8910.0 | nM | 5.05 |
| CHEMBL1325640 | — | EC50 | = | 9060.0 | nM | 5.04 |
| CHEMBL1599800 | — | EC50 | = | 9080.0 | nM | 5.04 |