Assay Detail
Functional
CHEMBL1738443
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR analysis of inhibitors of TNFa specific NF-kB induction - Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1575, AID1578, AID1852, AID2335, AID2337, AID2801]
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 20 | 5.17 | 5.88 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1419822 | — | — | 1 | 5.88 |
| CHEMBL1331314 | — | — | 1 | 5.48 |
| CHEMBL1452157 | — | — | 1 | 5.28 |
| CHEMBL1444568 | — | — | 1 | 5.25 |
| CHEMBL1519375 | — | — | 1 | 5.07 |
| CHEMBL1336829 | — | — | 1 | 4.88 |
| CHEMBL1468879 | — | — | 1 | 4.78 |
| CHEMBL1562608 | — | — | 1 | 4.77 |
| CHEMBL1603938 | — | — | 1 | - |
| CHEMBL1567543 | — | — | 1 | - |
| CHEMBL1332003 | — | — | 1 | - |
| CHEMBL1448844 | — | — | 1 | - |
| CHEMBL1345225 | — | — | 1 | - |
| CHEMBL1491481 | — | — | 1 | - |
| CHEMBL1412853 | — | — | 1 | - |
| CHEMBL1305184 | — | — | 1 | - |
| CHEMBL1595049 | — | — | 1 | - |
| CHEMBL1382232 | — | — | 1 | - |
| CHEMBL1299367 | — | — | 1 | - |
| CHEMBL1386167 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1419822 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1331314 | — | IC50 | = | 3310.0 | nM | 5.48 |
| CHEMBL1452157 | — | IC50 | = | 5210.0 | nM | 5.28 |
| CHEMBL1444568 | — | IC50 | = | 5690.0 | nM | 5.25 |
| CHEMBL1519375 | — | IC50 | = | 8490.0 | nM | 5.07 |
| CHEMBL1336829 | — | IC50 | = | 13100.0 | nM | 4.88 |
| CHEMBL1468879 | — | IC50 | = | 16800.0 | nM | 4.78 |
| CHEMBL1562608 | — | IC50 | = | 16900.0 | nM | 4.77 |
| CHEMBL1603938 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1567543 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1332003 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1448844 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1345225 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1491481 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1412853 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1305184 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1595049 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1382232 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1299367 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL1386167 | — | IC50 | > | 20000.0 | nM | - |