Assay Detail
Functional
CHEMBL1738480
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR Analysis of Selective Antagonists of GPR55 using an Image-Based Assay - Set 4. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2013, AID2026]
68
Total Activities
67
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 68 | 5.09 | 6.58 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1310336 | — | — | 1 | 6.58 |
| CHEMBL1484306 | — | — | 1 | 6.28 |
| CHEMBL1736438 | — | — | 1 | 5.75 |
| CHEMBL1704084 | — | — | 1 | 5.57 |
| CHEMBL1443900 | — | — | 1 | 5.53 |
| CHEMBL1730076 | — | — | 1 | 5.45 |
| CHEMBL1542448 | — | — | 1 | 5.40 |
| CHEMBL1730381 | — | — | 1 | 5.39 |
| CHEMBL1386647 | — | — | 1 | 5.38 |
| CHEMBL1402210 | — | — | 1 | 5.33 |
| CHEMBL1718220 | — | — | 1 | 5.28 |
| CHEMBL1725618 | — | — | 1 | 5.27 |
| CHEMBL1534425 | — | — | 1 | 5.24 |
| CHEMBL1717402 | — | — | 1 | 5.23 |
| CHEMBL1720072 | — | — | 1 | 5.23 |
| CHEMBL1722450 | — | — | 1 | 5.21 |
| CHEMBL1698983 | — | — | 1 | 5.16 |
| CHEMBL1719423 | — | — | 1 | 5.12 |
| CHEMBL1382214 | — | — | 1 | 5.11 |
| CHEMBL1411573 | — | — | 1 | 5.09 |
| CHEMBL1698745 | — | — | 1 | 5.09 |
| CHEMBL1718537 | — | — | 1 | 5.03 |
| CHEMBL1729479 | — | — | 1 | 5.02 |
| CHEMBL1721827 | — | — | 1 | 4.97 |
| CHEMBL1542604 | — | — | 2 | 4.96 |
| CHEMBL1727053 | — | — | 1 | 4.93 |
| CHEMBL1703285 | — | — | 1 | 4.89 |
| CHEMBL1703896 | — | — | 1 | 4.88 |
| CHEMBL1430124 | — | — | 1 | 4.86 |
| CHEMBL1698243 | — | — | 1 | 4.81 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1310336 | — | IC50 | = | 263.0 | nM | 6.58 |
| CHEMBL1484306 | — | IC50 | = | 527.0 | nM | 6.28 |
| CHEMBL1736438 | — | IC50 | = | 1770.0 | nM | 5.75 |
| CHEMBL1704084 | — | IC50 | = | 2700.0 | nM | 5.57 |
| CHEMBL1443900 | — | IC50 | = | 2950.0 | nM | 5.53 |
| CHEMBL1730076 | — | IC50 | = | 3560.0 | nM | 5.45 |
| CHEMBL1542448 | — | IC50 | = | 3950.0 | nM | 5.40 |
| CHEMBL1730381 | — | IC50 | = | 4100.0 | nM | 5.39 |
| CHEMBL1386647 | — | IC50 | = | 4130.0 | nM | 5.38 |
| CHEMBL1402210 | — | IC50 | = | 4630.0 | nM | 5.33 |
| CHEMBL1718220 | — | IC50 | = | 5270.0 | nM | 5.28 |
| CHEMBL1725618 | — | IC50 | = | 5400.0 | nM | 5.27 |
| CHEMBL1534425 | — | IC50 | = | 5750.0 | nM | 5.24 |
| CHEMBL1717402 | — | IC50 | = | 5920.0 | nM | 5.23 |
| CHEMBL1720072 | — | IC50 | = | 5850.0 | nM | 5.23 |
| CHEMBL1722450 | — | IC50 | = | 6130.0 | nM | 5.21 |
| CHEMBL1698983 | — | IC50 | = | 6890.0 | nM | 5.16 |
| CHEMBL1719423 | — | IC50 | = | 7600.0 | nM | 5.12 |
| CHEMBL1382214 | — | IC50 | = | 7700.0 | nM | 5.11 |
| CHEMBL1698745 | — | IC50 | = | 8180.0 | nM | 5.09 |
| CHEMBL1411573 | — | IC50 | = | 8040.0 | nM | 5.09 |
| CHEMBL1718537 | — | IC50 | = | 9240.0 | nM | 5.03 |
| CHEMBL1729479 | — | IC50 | = | 9550.0 | nM | 5.02 |
| CHEMBL1721827 | — | IC50 | = | 10600.0 | nM | 4.97 |
| CHEMBL1542604 | — | IC50 | = | 10900.0 | nM | 4.96 |
| CHEMBL1727053 | — | IC50 | = | 11700.0 | nM | 4.93 |
| CHEMBL1703285 | — | IC50 | = | 13000.0 | nM | 4.89 |
| CHEMBL1703896 | — | IC50 | = | 13100.0 | nM | 4.88 |
| CHEMBL1542604 | — | IC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL1430124 | — | IC50 | = | 13700.0 | nM | 4.86 |
| CHEMBL1698243 | — | IC50 | = | 15600.0 | nM | 4.81 |
| CHEMBL1703772 | — | IC50 | = | 17400.0 | nM | 4.76 |
| CHEMBL1708243 | — | IC50 | = | 18400.0 | nM | 4.74 |
| CHEMBL1481494 | — | IC50 | = | 18200.0 | nM | 4.74 |
| CHEMBL1734939 | — | IC50 | = | 19200.0 | nM | 4.72 |
| CHEMBL1726224 | — | IC50 | = | 19200.0 | nM | 4.72 |
| CHEMBL1715275 | — | IC50 | = | 21500.0 | nM | 4.67 |
| CHEMBL1701998 | — | IC50 | = | 21400.0 | nM | 4.67 |
| CHEMBL1710129 | — | IC50 | = | 22700.0 | nM | 4.64 |
| CHEMBL1586567 | — | IC50 | = | 28300.0 | nM | 4.55 |
| CHEMBL1727434 | — | IC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL1733320 | — | IC50 | = | 29000.0 | nM | 4.54 |
| CHEMBL1705660 | — | IC50 | = | 29700.0 | nM | 4.53 |
| CHEMBL1725686 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1416169 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1305795 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1705807 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1729109 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1728454 | — | IC50 | > | 32000.0 | nM | - |
| CHEMBL1726562 | — | IC50 | > | 32000.0 | nM | - |