Assay Detail
Functional
CHEMBL1738495
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of uHTS for inhibitors of Sentrin-specific protease 7 (SENP7) using a Luminescent assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID434973, AID434986]
704
Total Activities
704
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 704 | 5.18 | 6.45 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3196451 | — | — | 1 | 6.45 |
| CHEMBL281980 | — | — | 1 | 6.16 |
| CHEMBL3191962 | — | — | 1 | 6.12 |
| CHEMBL1402456 | — | — | 1 | 6.12 |
| CHEMBL1421255 | — | — | 1 | 6.10 |
| CHEMBL1506796 | — | — | 1 | 6.10 |
| CHEMBL1542328 | — | — | 1 | 6.07 |
| CHEMBL1967857 | — | — | 1 | 6.06 |
| CHEMBL1475128 | — | — | 1 | 6.03 |
| CHEMBL1418096 | — | — | 1 | 6.02 |
| CHEMBL3195102 | — | — | 1 | 6.00 |
| CHEMBL1449923 | — | — | 1 | 5.99 |
| CHEMBL595840 | — | — | 1 | 5.94 |
| CHEMBL1988780 | — | — | 1 | 5.91 |
| CHEMBL1417815 | — | — | 1 | 5.87 |
| CHEMBL1521051 | — | — | 1 | 5.84 |
| CHEMBL1380580 | — | — | 1 | 5.82 |
| CHEMBL3190318 | — | — | 1 | 5.80 |
| CHEMBL3210574 | — | — | 1 | 5.79 |
| CHEMBL1584379 | — | — | 1 | 5.79 |
| CHEMBL1498118 | — | — | 1 | 5.78 |
| CHEMBL205040 | — | — | 1 | 5.78 |
| CHEMBL1515340 | — | — | 1 | 5.77 |
| CHEMBL1477061 | — | — | 1 | 5.76 |
| CHEMBL1718258 | — | — | 1 | 5.76 |
| CHEMBL1705186 | — | — | 1 | 5.76 |
| CHEMBL1480814 | — | — | 1 | 5.75 |
| CHEMBL1301243 | — | — | 1 | 5.75 |
| CHEMBL1479657 | — | — | 1 | 5.73 |
| CHEMBL340701 | — | — | 1 | 5.72 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3196451 | — | IC50 | = | 359.0 | nM | 6.45 |
| CHEMBL281980 | — | IC50 | = | 696.0 | nM | 6.16 |
| CHEMBL3191962 | — | IC50 | = | 757.0 | nM | 6.12 |
| CHEMBL1402456 | — | IC50 | = | 750.0 | nM | 6.12 |
| CHEMBL1506796 | — | IC50 | = | 797.0 | nM | 6.10 |
| CHEMBL1421255 | — | IC50 | = | 788.0 | nM | 6.10 |
| CHEMBL1542328 | — | IC50 | = | 857.0 | nM | 6.07 |
| CHEMBL1967857 | — | IC50 | = | 863.0 | nM | 6.06 |
| CHEMBL1475128 | — | IC50 | = | 938.0 | nM | 6.03 |
| CHEMBL1418096 | — | IC50 | = | 955.0 | nM | 6.02 |
| CHEMBL3195102 | — | IC50 | = | 1010.0 | nM | 6.00 |
| CHEMBL1449923 | — | IC50 | = | 1020.0 | nM | 5.99 |
| CHEMBL595840 | — | IC50 | = | 1140.0 | nM | 5.94 |
| CHEMBL1988780 | — | IC50 | = | 1220.0 | nM | 5.91 |
| CHEMBL1417815 | — | IC50 | = | 1360.0 | nM | 5.87 |
| CHEMBL1521051 | — | IC50 | = | 1460.0 | nM | 5.84 |
| CHEMBL1380580 | — | IC50 | = | 1510.0 | nM | 5.82 |
| CHEMBL3190318 | — | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL1584379 | — | IC50 | = | 1640.0 | nM | 5.79 |
| CHEMBL3210574 | — | IC50 | = | 1640.0 | nM | 5.79 |
| CHEMBL1498118 | — | IC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL205040 | — | IC50 | = | 1670.0 | nM | 5.78 |
| CHEMBL1515340 | — | IC50 | = | 1690.0 | nM | 5.77 |
| CHEMBL1718258 | — | IC50 | = | 1730.0 | nM | 5.76 |
| CHEMBL1705186 | — | IC50 | = | 1750.0 | nM | 5.76 |
| CHEMBL1477061 | — | IC50 | = | 1740.0 | nM | 5.76 |
| CHEMBL1480814 | — | IC50 | = | 1780.0 | nM | 5.75 |
| CHEMBL1301243 | — | IC50 | = | 1790.0 | nM | 5.75 |
| CHEMBL1479657 | — | IC50 | = | 1850.0 | nM | 5.73 |
| CHEMBL1469807 | — | IC50 | = | 1890.0 | nM | 5.72 |
| CHEMBL340701 | — | IC50 | = | 1900.0 | nM | 5.72 |
| CHEMBL1379054 | — | IC50 | = | 1940.0 | nM | 5.71 |
| CHEMBL1890591 | — | IC50 | = | 1940.0 | nM | 5.71 |
| CHEMBL1712864 | — | IC50 | = | 1960.0 | nM | 5.71 |
| CHEMBL3194361 | — | IC50 | = | 1990.0 | nM | 5.70 |
| CHEMBL1998302 | — | IC50 | = | 2060.0 | nM | 5.69 |
| CHEMBL1504125 | — | IC50 | = | 2070.0 | nM | 5.68 |
| CHEMBL1349748 | — | IC50 | = | 2110.0 | nM | 5.68 |
| CHEMBL1544489 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL3198635 | — | IC50 | = | 2150.0 | nM | 5.67 |
| CHEMBL1582654 | — | IC50 | = | 2160.0 | nM | 5.67 |
| CHEMBL1321391 | — | IC50 | = | 2160.0 | nM | 5.67 |
| CHEMBL1532928 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL3196057 | — | IC50 | = | 2170.0 | nM | 5.66 |
| CHEMBL1707033 | — | IC50 | = | 2190.0 | nM | 5.66 |
| CHEMBL1719113 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL1339228 | — | IC50 | = | 2230.0 | nM | 5.65 |
| CHEMBL1604550 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL1438722 | — | IC50 | = | 2360.0 | nM | 5.63 |
| CHEMBL1303887 | — | IC50 | = | 2360.0 | nM | 5.63 |