Assay Detail
Functional
CHEMBL1738513
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response confirmation of small molecule activators of the apoptotic arm of the Unfolded Protein response via a luminescent-based reporter assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID449763, AID449771]
674
Total Activities
674
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 674 | 5.01 | 6.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1604863 | — | — | 1 | 6.38 |
| CHEMBL528694 | — | — | 1 | 6.19 |
| CHEMBL1550076 | — | — | 1 | 6.12 |
| CHEMBL1419414 | — | — | 1 | 6.09 |
| CHEMBL1725397 | — | — | 1 | 6.09 |
| CHEMBL319244 | CAFFEIC ACID PHENETHYL ESTER | — | 1 | 6.05 |
| CHEMBL1537810 | — | — | 1 | 6.04 |
| CHEMBL1335068 | — | — | 1 | 6.01 |
| CHEMBL1522618 | — | — | 1 | 5.97 |
| CHEMBL1991234 | — | — | 1 | 5.96 |
| CHEMBL2003964 | — | — | 1 | 5.91 |
| CHEMBL1533823 | — | — | 1 | 5.89 |
| CHEMBL3197092 | — | — | 1 | 5.88 |
| CHEMBL1987060 | — | — | 1 | 5.87 |
| CHEMBL1528581 | — | — | 1 | 5.87 |
| CHEMBL1444114 | — | — | 1 | 5.86 |
| CHEMBL1419335 | — | — | 1 | 5.81 |
| CHEMBL1580083 | — | — | 1 | 5.81 |
| CHEMBL1480798 | — | — | 1 | 5.81 |
| CHEMBL1378931 | — | — | 1 | 5.79 |
| CHEMBL546170 | — | — | 1 | 5.78 |
| CHEMBL1422161 | — | — | 1 | 5.75 |
| CHEMBL3190220 | — | — | 1 | 5.65 |
| CHEMBL1984876 | — | — | 1 | 5.63 |
| CHEMBL3109023 | — | — | 1 | 5.63 |
| CHEMBL3195898 | — | — | 1 | 5.62 |
| CHEMBL1544633 | — | — | 1 | 5.61 |
| CHEMBL1987579 | — | — | 1 | 5.60 |
| CHEMBL455284 | — | — | 1 | 5.60 |
| CHEMBL1567827 | — | — | 1 | 5.58 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1604863 | — | EC50 | = | 420.0 | nM | 6.38 |
| CHEMBL528694 | — | EC50 | = | 640.0 | nM | 6.19 |
| CHEMBL1550076 | — | EC50 | = | 750.0 | nM | 6.12 |
| CHEMBL1419414 | — | EC50 | = | 820.0 | nM | 6.09 |
| CHEMBL1725397 | — | EC50 | = | 810.0 | nM | 6.09 |
| CHEMBL319244 | CAFFEIC ACID PHENETHYL ESTER | EC50 | = | 890.0 | nM | 6.05 |
| CHEMBL1537810 | — | EC50 | = | 910.0 | nM | 6.04 |
| CHEMBL1335068 | — | EC50 | = | 980.0 | nM | 6.01 |
| CHEMBL1522618 | — | EC50 | = | 1080.0 | nM | 5.97 |
| CHEMBL1991234 | — | EC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL2003964 | — | EC50 | = | 1230.0 | nM | 5.91 |
| CHEMBL1533823 | — | EC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL3197092 | — | EC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1987060 | — | EC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL1528581 | — | EC50 | = | 1340.0 | nM | 5.87 |
| CHEMBL1444114 | — | EC50 | = | 1380.0 | nM | 5.86 |
| CHEMBL1580083 | — | EC50 | = | 1540.0 | nM | 5.81 |
| CHEMBL1480798 | — | EC50 | = | 1560.0 | nM | 5.81 |
| CHEMBL1419335 | — | EC50 | = | 1550.0 | nM | 5.81 |
| CHEMBL1378931 | — | EC50 | = | 1640.0 | nM | 5.79 |
| CHEMBL546170 | — | EC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL1422161 | — | EC50 | = | 1760.0 | nM | 5.75 |
| CHEMBL3190220 | — | EC50 | = | 2220.0 | nM | 5.65 |
| CHEMBL1984876 | — | EC50 | = | 2360.0 | nM | 5.63 |
| CHEMBL3109023 | — | EC50 | = | 2360.0 | nM | 5.63 |
| CHEMBL3195898 | — | EC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL1544633 | — | EC50 | = | 2480.0 | nM | 5.61 |
| CHEMBL1987579 | — | EC50 | = | 2510.0 | nM | 5.60 |
| CHEMBL455284 | — | EC50 | = | 2500.0 | nM | 5.60 |
| CHEMBL1567827 | — | EC50 | = | 2610.0 | nM | 5.58 |
| CHEMBL1564403 | — | EC50 | = | 2740.0 | nM | 5.56 |
| CHEMBL1544797 | — | EC50 | = | 2750.0 | nM | 5.56 |
| CHEMBL1987938 | — | EC50 | = | 2820.0 | nM | 5.55 |
| CHEMBL3196324 | — | EC50 | = | 2880.0 | nM | 5.54 |
| CHEMBL3208035 | — | EC50 | = | 2930.0 | nM | 5.53 |
| CHEMBL3192900 | — | EC50 | = | 2930.0 | nM | 5.53 |
| CHEMBL3192188 | — | EC50 | = | 3010.0 | nM | 5.52 |
| CHEMBL1342821 | — | EC50 | = | 3190.0 | nM | 5.50 |
| CHEMBL2094567 | — | EC50 | = | 3260.0 | nM | 5.49 |
| CHEMBL1976317 | — | EC50 | = | 3260.0 | nM | 5.49 |
| CHEMBL2094484 | — | EC50 | = | 3220.0 | nM | 5.49 |
| CHEMBL1423597 | — | EC50 | = | 3230.0 | nM | 5.49 |
| CHEMBL2003511 | — | EC50 | = | 3340.0 | nM | 5.48 |
| CHEMBL428064 | — | EC50 | = | 3420.0 | nM | 5.47 |
| CHEMBL391123 | — | EC50 | = | 3360.0 | nM | 5.47 |
| CHEMBL1563861 | — | EC50 | = | 3480.0 | nM | 5.46 |
| CHEMBL1321754 | — | EC50 | = | 3530.0 | nM | 5.45 |
| CHEMBL3199006 | — | EC50 | = | 3640.0 | nM | 5.44 |
| CHEMBL1597580 | — | EC50 | = | 3650.0 | nM | 5.44 |
| CHEMBL1300836 | — | EC50 | = | 3600.0 | nM | 5.44 |