Assay Detail
Functional
CHEMBL1738601
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR analysis of agonists of the Cannabinoid Receptor 2 using an Image-Based Assay. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID2013, AID2026]
38
Total Activities
38
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 38 | 4.52 | 4.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1460039 | — | — | 1 | 4.52 |
| CHEMBL1310336 | — | — | 1 | - |
| CHEMBL1421591 | — | — | 1 | - |
| CHEMBL1578189 | — | — | 1 | - |
| CHEMBL394883 | — | — | 1 | - |
| CHEMBL1431310 | — | — | 1 | - |
| CHEMBL1354041 | — | — | 1 | - |
| CHEMBL1448070 | — | — | 1 | - |
| CHEMBL1613157 | — | — | 1 | - |
| CHEMBL1466203 | — | — | 1 | - |
| CHEMBL1445966 | — | — | 1 | - |
| CHEMBL1572633 | — | — | 1 | - |
| CHEMBL1545109 | — | — | 1 | - |
| CHEMBL1581985 | — | — | 1 | - |
| CHEMBL1611658 | — | — | 1 | - |
| CHEMBL1582765 | — | — | 1 | - |
| CHEMBL1366039 | — | — | 1 | - |
| CHEMBL1410009 | — | — | 1 | - |
| CHEMBL1464477 | — | — | 1 | - |
| CHEMBL1498988 | — | — | 1 | - |
| CHEMBL1431953 | — | — | 1 | - |
| CHEMBL1411212 | — | — | 1 | - |
| CHEMBL1420800 | — | — | 1 | - |
| CHEMBL1549881 | — | — | 1 | - |
| CHEMBL1429129 | — | — | 1 | - |
| CHEMBL1468612 | — | — | 1 | - |
| CHEMBL1542168 | — | — | 1 | - |
| CHEMBL1567371 | — | — | 1 | - |
| CHEMBL1402920 | — | — | 1 | - |
| CHEMBL1575373 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1460039 | — | EC50 | = | 30200.0 | nM | 4.52 |
| CHEMBL1578189 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1572633 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1445966 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1466203 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1613157 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1448070 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1354041 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1431310 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL394883 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1545109 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1421591 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1507657 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1546161 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1386881 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1441155 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1484306 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1452959 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1420151 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1507172 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1411212 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1575373 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1402920 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1567371 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1542168 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1468612 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1429129 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1549881 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1420800 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1581985 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1431953 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1498988 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1464477 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1410009 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1366039 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1310336 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1582765 | — | EC50 | > | 32000.0 | nM | - |
| CHEMBL1611658 | — | EC50 | > | 32000.0 | nM | - |