Assay Detail
Functional
CHEMBL1738611
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose Response confirmation of APOBEC3A DNA Deaminase Inhibitors via a A3G counterscreen. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID493011, AID493024]
448
Total Activities
448
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
DNA dC->dU-editing enzyme APOBEC-3G (CHEMBL1741217) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 448 | 5.18 | 6.09 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3196851 | — | — | 1 | 6.09 |
| CHEMBL1362702 | — | — | 1 | 5.95 |
| CHEMBL3207528 | — | — | 1 | 5.90 |
| CHEMBL1342158 | — | — | 1 | 5.89 |
| CHEMBL1379279 | — | — | 1 | 5.88 |
| CHEMBL1389035 | — | — | 1 | 5.88 |
| CHEMBL1341547 | — | — | 1 | 5.85 |
| CHEMBL1501432 | — | — | 1 | 5.83 |
| CHEMBL225852 | GLAUCINE METHIODIDE | — | 1 | 5.78 |
| CHEMBL1377153 | — | — | 1 | 5.78 |
| CHEMBL1551307 | — | — | 1 | 5.76 |
| CHEMBL1706030 | — | — | 1 | 5.76 |
| CHEMBL1466065 | — | — | 1 | 5.74 |
| CHEMBL1510800 | — | — | 1 | 5.74 |
| CHEMBL1375102 | — | — | 1 | 5.72 |
| CHEMBL1577127 | — | — | 1 | 5.72 |
| CHEMBL1586607 | — | — | 1 | 5.72 |
| CHEMBL1732874 | — | — | 1 | 5.71 |
| CHEMBL1704847 | — | — | 1 | 5.71 |
| CHEMBL1519228 | — | — | 1 | 5.71 |
| CHEMBL1389793 | — | — | 1 | 5.70 |
| CHEMBL1575698 | — | — | 1 | 5.70 |
| CHEMBL1328041 | — | — | 1 | 5.70 |
| CHEMBL1543727 | — | — | 1 | 5.69 |
| CHEMBL1536626 | — | — | 1 | 5.68 |
| CHEMBL1408132 | — | — | 1 | 5.68 |
| CHEMBL1361245 | — | — | 1 | 5.68 |
| CHEMBL1698738 | — | — | 1 | 5.66 |
| CHEMBL1465029 | — | — | 1 | 5.66 |
| CHEMBL589421 | — | — | 1 | 5.66 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3196851 | — | IC50 | = | 814.0 | nM | 6.09 |
| CHEMBL1362702 | — | IC50 | = | 1120.0 | nM | 5.95 |
| CHEMBL3207528 | — | IC50 | = | 1260.0 | nM | 5.90 |
| CHEMBL1342158 | — | IC50 | = | 1290.0 | nM | 5.89 |
| CHEMBL1379279 | — | IC50 | = | 1310.0 | nM | 5.88 |
| CHEMBL1389035 | — | IC50 | = | 1320.0 | nM | 5.88 |
| CHEMBL1341547 | — | IC50 | = | 1420.0 | nM | 5.85 |
| CHEMBL1501432 | — | IC50 | = | 1470.0 | nM | 5.83 |
| CHEMBL1377153 | — | IC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL225852 | GLAUCINE METHIODIDE | IC50 | = | 1660.0 | nM | 5.78 |
| CHEMBL1706030 | — | IC50 | = | 1750.0 | nM | 5.76 |
| CHEMBL1551307 | — | IC50 | = | 1720.0 | nM | 5.76 |
| CHEMBL1510800 | — | IC50 | = | 1810.0 | nM | 5.74 |
| CHEMBL1466065 | — | IC50 | = | 1810.0 | nM | 5.74 |
| CHEMBL1577127 | — | IC50 | = | 1920.0 | nM | 5.72 |
| CHEMBL1375102 | — | IC50 | = | 1890.0 | nM | 5.72 |
| CHEMBL1586607 | — | IC50 | = | 1920.0 | nM | 5.72 |
| CHEMBL1732874 | — | IC50 | = | 1950.0 | nM | 5.71 |
| CHEMBL1704847 | — | IC50 | = | 1930.0 | nM | 5.71 |
| CHEMBL1519228 | — | IC50 | = | 1950.0 | nM | 5.71 |
| CHEMBL1575698 | — | IC50 | = | 2010.0 | nM | 5.70 |
| CHEMBL1389793 | — | IC50 | = | 1990.0 | nM | 5.70 |
| CHEMBL1328041 | — | IC50 | = | 2020.0 | nM | 5.70 |
| CHEMBL1543727 | — | IC50 | = | 2040.0 | nM | 5.69 |
| CHEMBL1361245 | — | IC50 | = | 2090.0 | nM | 5.68 |
| CHEMBL1536626 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL1408132 | — | IC50 | = | 2090.0 | nM | 5.68 |
| CHEMBL1338153 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL589421 | — | IC50 | = | 2170.0 | nM | 5.66 |
| CHEMBL1465029 | — | IC50 | = | 2190.0 | nM | 5.66 |
| CHEMBL1698738 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL1362088 | — | IC50 | = | 2240.0 | nM | 5.65 |
| CHEMBL1465047 | — | IC50 | = | 2260.0 | nM | 5.65 |
| CHEMBL1448452 | — | IC50 | = | 2230.0 | nM | 5.65 |
| CHEMBL1480280 | — | IC50 | = | 2220.0 | nM | 5.65 |
| CHEMBL1387510 | — | IC50 | = | 2240.0 | nM | 5.65 |
| CHEMBL1485727 | — | IC50 | = | 2310.0 | nM | 5.64 |
| CHEMBL1443664 | — | IC50 | = | 2290.0 | nM | 5.64 |
| CHEMBL1499690 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL1355123 | — | IC50 | = | 2300.0 | nM | 5.64 |
| CHEMBL1711351 | — | IC50 | = | 2270.0 | nM | 5.64 |
| CHEMBL3211324 | — | IC50 | = | 2350.0 | nM | 5.63 |
| CHEMBL1558595 | — | IC50 | = | 2360.0 | nM | 5.63 |
| CHEMBL1504638 | — | IC50 | = | 2420.0 | nM | 5.62 |
| CHEMBL1580846 | — | IC50 | = | 2410.0 | nM | 5.62 |
| CHEMBL1419432 | — | IC50 | = | 2410.0 | nM | 5.62 |
| CHEMBL1340231 | — | IC50 | = | 2420.0 | nM | 5.62 |
| CHEMBL1423563 | — | IC50 | = | 2410.0 | nM | 5.62 |
| CHEMBL1560104 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL1585158 | — | IC50 | = | 2440.0 | nM | 5.61 |