Assay Detail
Binding
CHEMBL1763569
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of CK1delta at 1 uM relative to control
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Discovery of triazine-benzimidazoles as selective inhibitors of mTOR.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 4.40 | 4.40 |
| Inhibition | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1615182 | — | — | 1 | 4.40 |
| CHEMBL1762782 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1615182 | — | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL1762782 | — | Inhibition | = | 90.0 | % | - |