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Assay Detail

CHEMBL1775561

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Zaire ebolavirus expressing enhanced GFP in Vero 76 cells after 48 hrs by standard Plaque assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Zaire ebolavirus
Cell Type Vero
Confidence 1 — Organism
Curated By Autocuration

Target

Ebolavirus (CHEMBL4434621)
Type ORGANISM
Organism Ebolavirus

Publication

A chemotype that inhibits three unrelated pathogenic targets: the botulinum neurotoxin serotype A light chain, P. falciparum malaria, and the Ebola filovirus.
Opsenica I, Burnett JC, Gussio R, Opsenica D, Todorović N, Lanteri CA, Sciotti RJ, Gettayacamin M, Basilico N, Taramelli D, Nuss JE, Wanner L, Panchal RG, Solaja BA, Bavari S.
J Med Chem (2011) 54 : 1157 -1169
PubMed 21265542 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.40 5.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1773165 1 5.60
CHEMBL1773160 1 5.30
CHEMBL1773163 1 5.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1773165 IC50 = 2500.0 nM 5.60
CHEMBL1773160 IC50 = 5000.0 nM 5.30
CHEMBL1773163 IC50 = 5000.0 nM 5.30