Assay Detail
Binding
CHEMBL1780744
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to guinea pig CRTh2 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Chemoattractant receptor-homologous molecule expressed on Th2 cells (CHEMBL1075058) ↗| Type | SINGLE PROTEIN |
| Organism | Cavia porcellus |
Publication
Switching between agonists and antagonists at CRTh2 in a series of highly potent and selective biaryl phenoxyacetic acids.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.20 | 7.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1778639 | — | — | 1 | 7.20 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1778639 | — | IC50 | = | 63.0 | nM | 7.20 |