Assay Detail
Functional
CHEMBL1787357
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiproliferative activity against human HeLaS3 cells after 72 hrs
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HeLa S3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis and biological evaluation of boron peptide analogues of Belactosin C as proteasome inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.29 | 4.29 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL491636 | BELACTOSIN A | — | 1 | 4.29 |
| CHEMBL1783833 | BELACTOSIN C | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL491636 | BELACTOSIN A | IC50 | = | 51000.0 | nM | 4.29 |
| CHEMBL1783833 | BELACTOSIN C | IC50 | = | 200000.0 | nM | - |