Assay Detail
Functional
CHEMBL1794296
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for inhibitors of TLR9-MyD88 binding: Luminescence-based cell-based high throughput dose response assay to identify cytotoxic compounds using TLR9-MyD88 CHO cells. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504734, AID504750, AID540250, AID540251]
235
Total Activities
234
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | hamster |
| Cell Type | CHO |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 235 | 5.44 | 6.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1698608 | — | — | 1 | 6.96 |
| CHEMBL1566610 | — | — | 1 | 6.83 |
| CHEMBL1790039 | — | — | 1 | 6.74 |
| CHEMBL505670 | — | — | 1 | 6.35 |
| CHEMBL1574879 | — | — | 1 | 6.34 |
| CHEMBL1494120 | — | — | 1 | 6.33 |
| CHEMBL429095 | — | — | 1 | 6.32 |
| CHEMBL1362660 | — | — | 1 | 6.26 |
| CHEMBL1732235 | — | — | 1 | 6.25 |
| CHEMBL1704703 | — | — | 1 | 6.24 |
| CHEMBL1734503 | — | — | 1 | 6.22 |
| CHEMBL1712082 | — | — | 1 | 6.21 |
| CHEMBL131037 | — | — | 1 | 6.20 |
| CHEMBL1698008 | — | — | 1 | 6.13 |
| CHEMBL1699845 | — | — | 1 | 6.13 |
| CHEMBL1526855 | — | — | 1 | 6.10 |
| CHEMBL1704261 | — | — | 1 | 6.05 |
| CHEMBL508338 | THIMEROSAL | 3.0 | 1 | 6.04 |
| CHEMBL1701517 | — | — | 1 | 6.02 |
| CHEMBL1999049 | — | — | 1 | 6.02 |
| CHEMBL1865393 | — | — | 1 | 5.99 |
| CHEMBL1988416 | — | — | 1 | 5.99 |
| CHEMBL1342053 | — | — | 1 | 5.99 |
| CHEMBL1404578 | — | — | 1 | 5.98 |
| CHEMBL1361740 | — | — | 1 | 5.97 |
| CHEMBL1308404 | — | — | 1 | 5.95 |
| CHEMBL1499951 | — | — | 1 | 5.93 |
| CHEMBL1440300 | — | — | 1 | 5.93 |
| CHEMBL1460029 | — | — | 1 | 5.91 |
| CHEMBL1611182 | — | — | 1 | 5.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1698608 | — | IC50 | = | 110.02 | nM | 6.96 |
| CHEMBL1566610 | — | IC50 | = | 147.37 | nM | 6.83 |
| CHEMBL1790039 | — | IC50 | = | 180.65 | nM | 6.74 |
| CHEMBL505670 | — | IC50 | = | 447.5 | nM | 6.35 |
| CHEMBL1574879 | — | IC50 | = | 453.44 | nM | 6.34 |
| CHEMBL1494120 | — | IC50 | = | 463.4 | nM | 6.33 |
| CHEMBL429095 | — | IC50 | = | 479.38 | nM | 6.32 |
| CHEMBL1362660 | — | IC50 | = | 545.52 | nM | 6.26 |
| CHEMBL1732235 | — | IC50 | = | 558.01 | nM | 6.25 |
| CHEMBL1704703 | — | IC50 | = | 569.53 | nM | 6.24 |
| CHEMBL1734503 | — | IC50 | = | 597.44 | nM | 6.22 |
| CHEMBL1712082 | — | IC50 | = | 618.7 | nM | 6.21 |
| CHEMBL131037 | — | IC50 | = | 629.47 | nM | 6.20 |
| CHEMBL1699845 | — | IC50 | = | 738.11 | nM | 6.13 |
| CHEMBL1698008 | — | IC50 | = | 745.15 | nM | 6.13 |
| CHEMBL1526855 | — | IC50 | = | 801.9 | nM | 6.10 |
| CHEMBL1704261 | — | IC50 | = | 890.86 | nM | 6.05 |
| CHEMBL508338 | THIMEROSAL | IC50 | = | 921.0 | nM | 6.04 |
| CHEMBL1999049 | — | IC50 | = | 952.0 | nM | 6.02 |
| CHEMBL1701517 | — | IC50 | = | 959.0 | nM | 6.02 |
| CHEMBL1342053 | — | IC50 | = | 1032.0 | nM | 5.99 |
| CHEMBL1865393 | — | IC50 | = | 1034.0 | nM | 5.99 |
| CHEMBL1988416 | — | IC50 | = | 1030.0 | nM | 5.99 |
| CHEMBL1404578 | — | IC50 | = | 1048.0 | nM | 5.98 |
| CHEMBL1361740 | — | IC50 | = | 1080.0 | nM | 5.97 |
| CHEMBL1308404 | — | IC50 | = | 1130.0 | nM | 5.95 |
| CHEMBL1499951 | — | IC50 | = | 1182.0 | nM | 5.93 |
| CHEMBL1440300 | — | IC50 | = | 1178.0 | nM | 5.93 |
| CHEMBL1460029 | — | IC50 | = | 1218.0 | nM | 5.91 |
| CHEMBL1611182 | — | IC50 | = | 1273.0 | nM | 5.89 |
| CHEMBL1413680 | — | IC50 | = | 1295.0 | nM | 5.89 |
| CHEMBL1711514 | — | IC50 | = | 1335.0 | nM | 5.88 |
| CHEMBL1319867 | — | IC50 | = | 1364.0 | nM | 5.87 |
| CHEMBL1458022 | — | IC50 | = | 1385.0 | nM | 5.86 |
| CHEMBL1303810 | — | IC50 | = | 1457.0 | nM | 5.84 |
| CHEMBL601543 | — | IC50 | = | 1448.0 | nM | 5.84 |
| CHEMBL1303426 | — | IC50 | = | 1528.0 | nM | 5.82 |
| CHEMBL1343392 | — | IC50 | = | 1535.0 | nM | 5.81 |
| CHEMBL1497139 | — | IC50 | = | 1561.0 | nM | 5.81 |
| CHEMBL1555532 | — | IC50 | = | 1596.0 | nM | 5.80 |
| CHEMBL1710816 | — | IC50 | = | 1588.0 | nM | 5.80 |
| CHEMBL1723955 | — | IC50 | = | 1583.0 | nM | 5.80 |
| CHEMBL1543839 | — | IC50 | = | 1639.0 | nM | 5.79 |
| CHEMBL1427185 | — | IC50 | = | 1625.0 | nM | 5.79 |
| CHEMBL1585390 | — | IC50 | = | 1676.0 | nM | 5.78 |
| CHEMBL1301723 | — | IC50 | = | 1644.0 | nM | 5.78 |
| CHEMBL1567159 | — | IC50 | = | 1686.0 | nM | 5.77 |
| CHEMBL1351081 | — | IC50 | = | 1696.0 | nM | 5.77 |
| CHEMBL1711797 | — | IC50 | = | 1689.0 | nM | 5.77 |
| CHEMBL428064 | — | IC50 | = | 1769.0 | nM | 5.75 |