Assay Detail
Functional
CHEMBL1794407
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR VHR1 Fluorescent Assay for In Vitro dose response studies Set 3. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1654, AID1661, AID1878]
27
Total Activities
27
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Dual specificity protein phosphatase 3 (CHEMBL2635) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 27 | 4.83 | 6.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1892801 | — | — | 1 | 6.17 |
| CHEMBL1349451 | — | — | 1 | 5.44 |
| CHEMBL1882430 | — | — | 1 | 5.43 |
| CHEMBL1325709 | — | — | 1 | 5.43 |
| CHEMBL1390963 | — | — | 1 | 5.14 |
| CHEMBL1301776 | — | — | 1 | 4.94 |
| CHEMBL1576545 | — | — | 1 | 4.92 |
| CHEMBL1871792 | — | — | 1 | 4.92 |
| CHEMBL1867272 | — | — | 1 | 4.86 |
| CHEMBL1882306 | — | — | 1 | 4.81 |
| CHEMBL1333386 | — | — | 1 | 4.81 |
| CHEMBL1349331 | — | — | 1 | 4.74 |
| CHEMBL1901358 | — | — | 1 | 4.60 |
| CHEMBL1906065 | — | — | 1 | 4.44 |
| CHEMBL1866687 | — | — | 1 | 4.39 |
| CHEMBL446577 | — | — | 1 | 4.38 |
| CHEMBL1903660 | — | — | 1 | 4.31 |
| CHEMBL1872546 | — | — | 1 | 4.29 |
| CHEMBL1873104 | — | — | 1 | 4.24 |
| CHEMBL523954 | — | — | 1 | 4.24 |
| CHEMBL1899204 | — | — | 1 | - |
| CHEMBL1886697 | — | — | 1 | - |
| CHEMBL1882605 | — | — | 1 | - |
| CHEMBL1903677 | — | — | 1 | - |
| CHEMBL1896936 | — | — | 1 | - |
| CHEMBL1868126 | — | — | 1 | - |
| CHEMBL1865327 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1892801 | — | IC50 | = | 682.0 | nM | 6.17 |
| CHEMBL1349451 | — | IC50 | = | 3610.0 | nM | 5.44 |
| CHEMBL1882430 | — | IC50 | = | 3710.0 | nM | 5.43 |
| CHEMBL1325709 | — | IC50 | = | 3690.0 | nM | 5.43 |
| CHEMBL1390963 | — | IC50 | = | 7300.0 | nM | 5.14 |
| CHEMBL1301776 | — | IC50 | = | 11400.0 | nM | 4.94 |
| CHEMBL1576545 | — | IC50 | = | 12100.0 | nM | 4.92 |
| CHEMBL1871792 | — | IC50 | = | 12000.0 | nM | 4.92 |
| CHEMBL1867272 | — | IC50 | = | 13700.0 | nM | 4.86 |
| CHEMBL1882306 | — | IC50 | = | 15400.0 | nM | 4.81 |
| CHEMBL1333386 | — | IC50 | = | 15600.0 | nM | 4.81 |
| CHEMBL1349331 | — | IC50 | = | 18300.0 | nM | 4.74 |
| CHEMBL1901358 | — | IC50 | = | 25300.0 | nM | 4.60 |
| CHEMBL1906065 | — | IC50 | = | 36300.0 | nM | 4.44 |
| CHEMBL1866687 | — | IC50 | = | 40600.0 | nM | 4.39 |
| CHEMBL446577 | — | IC50 | = | 41900.0 | nM | 4.38 |
| CHEMBL1903660 | — | IC50 | = | 48700.0 | nM | 4.31 |
| CHEMBL1872546 | — | IC50 | = | 51700.0 | nM | 4.29 |
| CHEMBL1873104 | — | IC50 | = | 58200.0 | nM | 4.24 |
| CHEMBL523954 | — | IC50 | = | 57600.0 | nM | 4.24 |
| CHEMBL1899204 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1886697 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1882605 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1903677 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1896936 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1868126 | — | IC50 | > | 66000.0 | nM | - |
| CHEMBL1865327 | — | IC50 | > | 66000.0 | nM | - |