Assay Detail
Binding
CHEMBL1794438
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for inhibitors of TLR9-MyD88 binding: fluorescence-based cell-based high throughput dose response assay to identify non-selective inhibitors of the beta-lactamase enzyme (BLA). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504734, AID504750, AID540250, AID540251]
235
Total Activities
234
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 235 | 5.10 | 5.67 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3197908 | — | — | 1 | 5.67 |
| CHEMBL1418079 | — | — | 1 | 5.64 |
| CHEMBL1360031 | — | — | 1 | 5.63 |
| CHEMBL1520346 | — | — | 1 | 5.59 |
| CHEMBL1526126 | — | — | 1 | 5.58 |
| CHEMBL1899958 | — | — | 1 | 5.56 |
| CHEMBL1554784 | — | — | 1 | 5.54 |
| CHEMBL1991303 | — | — | 1 | 5.52 |
| CHEMBL1472131 | — | — | 1 | 5.51 |
| CHEMBL1315948 | — | — | 1 | 5.50 |
| CHEMBL1436864 | — | — | 1 | 5.49 |
| CHEMBL1491686 | — | — | 1 | 5.48 |
| CHEMBL1415985 | — | — | 1 | 5.46 |
| CHEMBL1446199 | — | — | 1 | 5.45 |
| CHEMBL1705527 | — | — | 1 | 5.44 |
| CHEMBL1508593 | — | — | 1 | 5.44 |
| CHEMBL1513846 | — | — | 1 | 5.44 |
| CHEMBL1417212 | — | — | 1 | 5.44 |
| CHEMBL1399957 | — | — | 1 | 5.43 |
| CHEMBL1578982 | — | — | 1 | 5.43 |
| CHEMBL1984244 | — | — | 1 | 5.43 |
| CHEMBL1470904 | — | — | 1 | 5.43 |
| CHEMBL1541918 | — | — | 1 | 5.43 |
| CHEMBL1458470 | — | — | 1 | 5.42 |
| CHEMBL1527994 | — | — | 1 | 5.42 |
| CHEMBL1500409 | — | — | 1 | 5.42 |
| CHEMBL1387110 | — | — | 1 | 5.41 |
| CHEMBL1340895 | — | — | 1 | 5.41 |
| CHEMBL1418428 | — | — | 1 | 5.41 |
| CHEMBL1390797 | — | — | 1 | 5.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3197908 | — | IC50 | = | 2129.0 | nM | 5.67 |
| CHEMBL1418079 | — | IC50 | = | 2270.0 | nM | 5.64 |
| CHEMBL1360031 | — | IC50 | = | 2366.0 | nM | 5.63 |
| CHEMBL1520346 | — | IC50 | = | 2560.0 | nM | 5.59 |
| CHEMBL1526126 | — | IC50 | = | 2639.0 | nM | 5.58 |
| CHEMBL1899958 | — | IC50 | = | 2744.0 | nM | 5.56 |
| CHEMBL1554784 | — | IC50 | = | 2919.0 | nM | 5.54 |
| CHEMBL1991303 | — | IC50 | = | 2995.0 | nM | 5.52 |
| CHEMBL1472131 | — | IC50 | = | 3071.0 | nM | 5.51 |
| CHEMBL1315948 | — | IC50 | = | 3124.0 | nM | 5.50 |
| CHEMBL1436864 | — | IC50 | = | 3211.0 | nM | 5.49 |
| CHEMBL1491686 | — | IC50 | = | 3320.0 | nM | 5.48 |
| CHEMBL1415985 | — | IC50 | = | 3479.0 | nM | 5.46 |
| CHEMBL1446199 | — | IC50 | = | 3518.0 | nM | 5.45 |
| CHEMBL1705527 | — | IC50 | = | 3598.0 | nM | 5.44 |
| CHEMBL1513846 | — | IC50 | = | 3661.0 | nM | 5.44 |
| CHEMBL1417212 | — | IC50 | = | 3616.0 | nM | 5.44 |
| CHEMBL1508593 | — | IC50 | = | 3667.0 | nM | 5.44 |
| CHEMBL1541918 | — | IC50 | = | 3730.0 | nM | 5.43 |
| CHEMBL1470904 | — | IC50 | = | 3698.0 | nM | 5.43 |
| CHEMBL1578982 | — | IC50 | = | 3732.0 | nM | 5.43 |
| CHEMBL1399957 | — | IC50 | = | 3685.0 | nM | 5.43 |
| CHEMBL1984244 | — | IC50 | = | 3709.0 | nM | 5.43 |
| CHEMBL1527994 | — | IC50 | = | 3823.0 | nM | 5.42 |
| CHEMBL1500409 | — | IC50 | = | 3850.0 | nM | 5.42 |
| CHEMBL1458470 | — | IC50 | = | 3785.0 | nM | 5.42 |
| CHEMBL1434843 | — | IC50 | = | 3875.0 | nM | 5.41 |
| CHEMBL1418428 | — | IC50 | = | 3901.0 | nM | 5.41 |
| CHEMBL1340895 | — | IC50 | = | 3924.0 | nM | 5.41 |
| CHEMBL1390797 | — | IC50 | = | 3855.0 | nM | 5.41 |
| CHEMBL1387110 | — | IC50 | = | 3934.0 | nM | 5.41 |
| CHEMBL432044 | — | IC50 | = | 3968.0 | nM | 5.40 |
| CHEMBL2005437 | — | IC50 | = | 4044.0 | nM | 5.39 |
| CHEMBL1573592 | — | IC50 | = | 4057.0 | nM | 5.39 |
| CHEMBL1964993 | — | IC50 | = | 4186.0 | nM | 5.38 |
| CHEMBL1459316 | — | IC50 | = | 4385.0 | nM | 5.36 |
| CHEMBL1583998 | — | IC50 | = | 4369.0 | nM | 5.36 |
| CHEMBL1726287 | — | IC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL1418162 | — | IC50 | = | 4497.0 | nM | 5.35 |
| CHEMBL1720248 | — | IC50 | = | 4504.0 | nM | 5.35 |
| CHEMBL1462613 | — | IC50 | = | 4440.0 | nM | 5.35 |
| CHEMBL1430995 | — | IC50 | = | 4592.0 | nM | 5.34 |
| CHEMBL1534390 | — | IC50 | = | 4583.0 | nM | 5.34 |
| CHEMBL61559 | — | IC50 | = | 4712.0 | nM | 5.33 |
| CHEMBL1479144 | — | IC50 | = | 4736.0 | nM | 5.33 |
| CHEMBL1999014 | — | IC50 | = | 4695.0 | nM | 5.33 |
| CHEMBL1585390 | — | IC50 | = | 4730.0 | nM | 5.33 |
| CHEMBL1301731 | — | IC50 | = | 4768.0 | nM | 5.32 |
| CHEMBL1725771 | — | IC50 | = | 4771.0 | nM | 5.32 |
| CHEMBL137913 | — | IC50 | = | 4770.0 | nM | 5.32 |