Assay Detail
Functional
CHEMBL1794498
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: SAR Analysis of small molecule inhibitors of Sentrin-specific protease 7 (SENP7) using a Luminescent assay - Set 2. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID434973, AID434986]
101
Total Activities
101
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 101 | 5.35 | 6.25 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1870914 | — | — | 1 | 6.25 |
| CHEMBL1316867 | — | — | 1 | 6.23 |
| CHEMBL1871228 | — | — | 1 | 6.01 |
| CHEMBL1869393 | — | — | 1 | 5.94 |
| CHEMBL1891206 | — | — | 1 | 5.92 |
| CHEMBL1302779 | — | — | 1 | 5.91 |
| CHEMBL1577231 | — | — | 1 | 5.87 |
| CHEMBL1319405 | — | — | 1 | 5.87 |
| CHEMBL1877777 | — | — | 1 | 5.86 |
| CHEMBL1866613 | — | — | 1 | 5.81 |
| CHEMBL1483649 | — | — | 1 | 5.78 |
| CHEMBL1553773 | — | — | 1 | 5.73 |
| CHEMBL1705186 | — | — | 1 | 5.73 |
| CHEMBL1868902 | — | — | 1 | 5.71 |
| CHEMBL1901952 | — | — | 1 | 5.68 |
| CHEMBL1904648 | — | — | 1 | 5.68 |
| CHEMBL1869506 | — | — | 1 | 5.68 |
| CHEMBL1903348 | — | — | 1 | 5.67 |
| CHEMBL1899989 | — | — | 1 | 5.65 |
| CHEMBL1333222 | — | — | 1 | 5.64 |
| CHEMBL1864747 | — | — | 1 | 5.57 |
| CHEMBL1868274 | — | — | 1 | 5.57 |
| CHEMBL1899595 | — | — | 1 | 5.57 |
| CHEMBL1886662 | — | — | 1 | 5.54 |
| CHEMBL1896263 | — | — | 1 | 5.48 |
| CHEMBL1871327 | — | — | 1 | 5.47 |
| CHEMBL1886317 | — | — | 1 | 5.38 |
| CHEMBL1896451 | — | — | 1 | 5.27 |
| CHEMBL1865625 | — | — | 1 | 5.23 |
| CHEMBL1884442 | — | — | 1 | 5.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1870914 | — | IC50 | = | 558.0 | nM | 6.25 |
| CHEMBL1316867 | — | IC50 | = | 589.0 | nM | 6.23 |
| CHEMBL1871228 | — | IC50 | = | 987.0 | nM | 6.01 |
| CHEMBL1869393 | — | IC50 | = | 1160.0 | nM | 5.94 |
| CHEMBL1891206 | — | IC50 | = | 1210.0 | nM | 5.92 |
| CHEMBL1302779 | — | IC50 | = | 1230.0 | nM | 5.91 |
| CHEMBL1577231 | — | IC50 | = | 1350.0 | nM | 5.87 |
| CHEMBL1319405 | — | IC50 | = | 1360.0 | nM | 5.87 |
| CHEMBL1877777 | — | IC50 | = | 1390.0 | nM | 5.86 |
| CHEMBL1866613 | — | IC50 | = | 1540.0 | nM | 5.81 |
| CHEMBL1483649 | — | IC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL1553773 | — | IC50 | = | 1870.0 | nM | 5.73 |
| CHEMBL1705186 | — | IC50 | = | 1850.0 | nM | 5.73 |
| CHEMBL1868902 | — | IC50 | = | 1960.0 | nM | 5.71 |
| CHEMBL1869506 | — | IC50 | = | 2080.0 | nM | 5.68 |
| CHEMBL1904648 | — | IC50 | = | 2090.0 | nM | 5.68 |
| CHEMBL1901952 | — | IC50 | = | 2080.0 | nM | 5.68 |
| CHEMBL1903348 | — | IC50 | = | 2130.0 | nM | 5.67 |
| CHEMBL1899989 | — | IC50 | = | 2220.0 | nM | 5.65 |
| CHEMBL1333222 | — | IC50 | = | 2310.0 | nM | 5.64 |
| CHEMBL1864747 | — | IC50 | = | 2710.0 | nM | 5.57 |
| CHEMBL1868274 | — | IC50 | = | 2670.0 | nM | 5.57 |
| CHEMBL1899595 | — | IC50 | = | 2700.0 | nM | 5.57 |
| CHEMBL1886662 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL1896263 | — | IC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL1871327 | — | IC50 | = | 3380.0 | nM | 5.47 |
| CHEMBL1886317 | — | IC50 | = | 4140.0 | nM | 5.38 |
| CHEMBL1896451 | — | IC50 | = | 5420.0 | nM | 5.27 |
| CHEMBL1865625 | — | IC50 | = | 5860.0 | nM | 5.23 |
| CHEMBL1884442 | — | IC50 | = | 6060.0 | nM | 5.22 |
| CHEMBL1882443 | — | IC50 | = | 6320.0 | nM | 5.20 |
| CHEMBL1564500 | — | IC50 | = | 7460.0 | nM | 5.13 |
| CHEMBL1878043 | — | IC50 | = | 7780.0 | nM | 5.11 |
| CHEMBL1902007 | — | IC50 | = | 8020.0 | nM | 5.10 |
| CHEMBL1887272 | — | IC50 | = | 8400.0 | nM | 5.08 |
| CHEMBL1365469 | — | IC50 | = | 8260.0 | nM | 5.08 |
| CHEMBL1878061 | — | IC50 | = | 10300.0 | nM | 4.99 |
| CHEMBL1898423 | — | IC50 | = | 11100.0 | nM | 4.96 |
| CHEMBL1872841 | — | IC50 | = | 12200.0 | nM | 4.91 |
| CHEMBL1897885 | — | IC50 | = | 14900.0 | nM | 4.83 |
| CHEMBL1874506 | — | IC50 | = | 19200.0 | nM | 4.72 |
| CHEMBL1883257 | — | IC50 | = | 29400.0 | nM | 4.53 |
| CHEMBL1896949 | — | IC50 | = | 34400.0 | nM | 4.46 |
| CHEMBL1413278 | — | IC50 | = | 43800.0 | nM | 4.36 |
| CHEMBL1874988 | — | IC50 | = | 72300.0 | nM | 4.14 |
| CHEMBL1899813 | — | IC50 | = | 88800.0 | nM | 4.05 |
| CHEMBL1890960 | — | IC50 | = | 95700.0 | nM | 4.02 |
| CHEMBL1886655 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1437840 | — | IC50 | > | 99000.0 | nM | - |
| CHEMBL1864230 | — | IC50 | > | 99000.0 | nM | - |