Assay Detail
Functional
CHEMBL1794508
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for inhibitors of the orphan nuclear receptor subfamily 0, group B, member 1 (DAX1; NR0B1): luminescence-based cell-based high throughput dose response assay to identify compounds that interfere with the UAS/Gal4 system and/or luciferase reporter. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID504766, AID504790]
242
Total Activities
242
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 242 | 5.22 | 6.74 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL98 | VORINOSTAT | 4.0 | 1 | 6.74 |
| CHEMBL1351761 | DINALINE | -1.0 | 1 | 6.59 |
| CHEMBL1488450 | — | — | 1 | 6.16 |
| CHEMBL1592550 | — | — | 1 | 5.99 |
| CHEMBL1557898 | — | — | 1 | 5.80 |
| CHEMBL1537451 | — | — | 1 | 5.72 |
| CHEMBL1485099 | — | — | 1 | 5.46 |
| CHEMBL1556370 | — | — | 1 | 4.61 |
| CHEMBL1470718 | — | — | 1 | 4.61 |
| CHEMBL3190167 | — | — | 1 | 4.33 |
| CHEMBL1486187 | — | — | 1 | 4.30 |
| CHEMBL1404302 | — | — | 1 | 4.29 |
| CHEMBL1542814 | — | — | 1 | 4.25 |
| CHEMBL1433231 | — | — | 1 | 4.18 |
| CHEMBL1885439 | — | — | 1 | - |
| CHEMBL1536643 | — | — | 1 | - |
| CHEMBL3199849 | — | — | 1 | - |
| CHEMBL1458054 | — | — | 1 | - |
| CHEMBL1299628 | — | — | 1 | - |
| CHEMBL1885548 | — | — | 1 | - |
| CHEMBL605752 | — | — | 1 | - |
| CHEMBL1533576 | — | — | 1 | - |
| CHEMBL1526696 | — | — | 1 | - |
| CHEMBL1967184 | — | — | 1 | - |
| CHEMBL1864101 | — | — | 1 | - |
| CHEMBL1604446 | — | — | 1 | - |
| CHEMBL1526666 | — | — | 1 | - |
| CHEMBL1698257 | — | — | 1 | - |
| CHEMBL16312 | 4'-METHOXYFLAVONE | — | 1 | - |
| CHEMBL1604097 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL98 | VORINOSTAT | IC50 | = | 183.11 | nM | 6.74 |
| CHEMBL1351761 | DINALINE | IC50 | = | 255.07 | nM | 6.59 |
| CHEMBL1488450 | — | IC50 | = | 695.37 | nM | 6.16 |
| CHEMBL1592550 | — | IC50 | = | 1036.0 | nM | 5.99 |
| CHEMBL1557898 | — | IC50 | = | 1586.0 | nM | 5.80 |
| CHEMBL1537451 | — | IC50 | = | 1910.0 | nM | 5.72 |
| CHEMBL1485099 | — | IC50 | = | 3473.0 | nM | 5.46 |
| CHEMBL1470718 | — | IC50 | = | 24702.0 | nM | 4.61 |
| CHEMBL1556370 | — | IC50 | = | 24602.0 | nM | 4.61 |
| CHEMBL3190167 | — | IC50 | = | 46947.0 | nM | 4.33 |
| CHEMBL1486187 | — | IC50 | = | 50374.0 | nM | 4.30 |
| CHEMBL1404302 | — | IC50 | = | 51744.0 | nM | 4.29 |
| CHEMBL1542814 | — | IC50 | = | 56055.0 | nM | 4.25 |
| CHEMBL1433231 | — | IC50 | = | 65247.0 | nM | 4.18 |
| CHEMBL1406761 | — | IC50 | > | 67493.0 | nM | - |
| CHEMBL1373715 | — | IC50 | > | 67529.0 | nM | - |
| CHEMBL1462180 | — | IC50 | > | 67481.0 | nM | - |
| CHEMBL3197401 | — | IC50 | > | 67499.0 | nM | - |
| CHEMBL1374578 | — | IC50 | > | 67534.0 | nM | - |
| CHEMBL1878128 | — | IC50 | > | 67541.0 | nM | - |
| CHEMBL1730712 | — | IC50 | > | 67568.0 | nM | - |
| CHEMBL1413278 | — | IC50 | > | 67504.0 | nM | - |
| CHEMBL1303248 | — | IC50 | > | 67574.0 | nM | - |
| CHEMBL1585571 | — | IC50 | > | 67547.0 | nM | - |
| CHEMBL1429314 | — | IC50 | > | 67481.0 | nM | - |
| CHEMBL1303246 | — | IC50 | > | 67554.0 | nM | - |
| CHEMBL1310006 | — | IC50 | > | 67491.0 | nM | - |
| CHEMBL1530924 | — | IC50 | > | 67506.0 | nM | - |
| CHEMBL1479907 | — | IC50 | > | 67527.0 | nM | - |
| CHEMBL1969590 | — | IC50 | > | 67547.0 | nM | - |
| CHEMBL3189729 | — | IC50 | > | 67547.0 | nM | - |
| CHEMBL1530910 | — | IC50 | > | 67528.0 | nM | - |
| CHEMBL1334807 | — | IC50 | > | 67541.0 | nM | - |
| CHEMBL1350621 | — | IC50 | > | 67581.0 | nM | - |
| CHEMBL1532144 | — | IC50 | > | 67536.0 | nM | - |
| CHEMBL1370549 | — | IC50 | > | 67541.0 | nM | - |
| CHEMBL1712486 | — | IC50 | > | 67541.0 | nM | - |
| CHEMBL1711986 | — | IC50 | > | 67554.0 | nM | - |
| CHEMBL1597768 | — | IC50 | > | 67602.0 | nM | - |
| CHEMBL1485549 | — | IC50 | > | 67537.0 | nM | - |
| CHEMBL1558980 | — | IC50 | > | 67506.0 | nM | - |
| CHEMBL16482 | — | IC50 | > | 67462.0 | nM | - |
| CHEMBL1879191 | — | IC50 | > | 67527.0 | nM | - |
| CHEMBL1711590 | — | IC50 | > | 67522.0 | nM | - |
| CHEMBL1586769 | — | IC50 | > | 67561.0 | nM | - |
| CHEMBL1730875 | — | IC50 | > | 67541.0 | nM | - |
| CHEMBL1469346 | — | IC50 | > | 67547.0 | nM | - |
| CHEMBL1532005 | — | IC50 | > | 67608.0 | nM | - |
| CHEMBL1303845 | — | IC50 | > | 67501.0 | nM | - |
| CHEMBL1711109 | — | IC50 | > | 67518.0 | nM | - |