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Assay Detail

CHEMBL1803176

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Functional
Antiviral activity against Cowpox virus Brighton infected in HFF cells assessed as reduction in plaque formation after 3 days
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Cowpox virus (Brighton Red)
Cell Type HFF
Confidence 1 — Organism
Curated By Autocuration

Publication

Synthesis, transport and antiviral activity of Ala-Ser and Val-Ser prodrugs of cidofovir.
Peterson LW, Kim JS, Kijek P, Mitchell S, Hilfinger J, Breitenbach J, Borysko K, Drach JC, Kashemirov BA, McKenna CE.
Bioorg Med Chem Lett (2011) 21 : 4045 -4049
PubMed 21641218 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.52 4.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5314375 CIDOFOVIR 4.0 1 4.52
CHEMBL392630 CYCLIC CIDOFOVIR 1 4.52
CHEMBL1802859 1 -
CHEMBL1802860 1 -
CHEMBL1802862 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5314375 CIDOFOVIR IC50 = 30000.0 nM 4.52
CHEMBL392630 CYCLIC CIDOFOVIR IC50 = 30000.0 nM 4.52
CHEMBL1802859 IC50 > 100000.0 nM -
CHEMBL1802860 IC50 > 100000.0 nM -
CHEMBL1802862 IC50 > 30000.0 nM -