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Assay Detail

CHEMBL1811512

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ADMET
Cytotoxicity against human HEK293T cells expressing AP-1 after 18 hrs by XTT assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type HEK-293T
Confidence 1 — Organism
Curated By Autocuration

Target

HEK-293T (CHEMBL3706568)
Type CELL-LINE
Organism Homo sapiens

Publication

Nothospondin, a new AP-1 inhibitory quassinoid from the Cameroonian plant Nothospondias staudtii.
Diyabalanage T, Ratnayake R, Wilson JA, Henrich CJ, Beutler JA, Colburn NH, McMahon JB, Gustafson KR.
Bioorg Med Chem Lett (2011) 21 : 4397 -4399
PubMed 21733691 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.00 5.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1807644 NOTHOSPONDIN 1 5.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1807644 NOTHOSPONDIN IC50 = 10000.0 nM 5.00