Assay Detail
Functional
CHEMBL1831791
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Cytotoxicity against human KB cells
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | KB |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Bioactive components from the heartwood of Pterocarpus santalinus.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 4.79 | 5.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL428647 | PACLITAXEL | 4.0 | 1 | 5.17 |
| CHEMBL1829657 | PTEROLINUS L | — | 1 | 4.76 |
| CHEMBL1613209 | CEAROIN | — | 1 | 4.45 |
| CHEMBL1829656 | PTEROLINUS K | — | 1 | - |
| CHEMBL1829658 | DALBERGIN | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL428647 | PACLITAXEL | IC50 | = | 6684.0 | nM | 5.17 |
| CHEMBL1829657 | PTEROLINUS L | IC50 | = | 17180.0 | nM | 4.76 |
| CHEMBL1613209 | CEAROIN | IC50 | = | 35330.0 | nM | 4.45 |
| CHEMBL1829656 | PTEROLINUS K | IC50 | > | 10.0 | ug.mL-1 | - |
| CHEMBL1829658 | DALBERGIN | IC50 | > | 10.0 | ug.mL-1 | - |