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Assay Detail

CHEMBL1839679

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Functional
Cytotoxicity against human PC3M cells by propidium iodide staining
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type PC-3M
Confidence 1 — Organism
Curated By Autocuration

Publication

Hydrazidomycins, cytotoxic alkylhydrazides from Streptomycesatratus.
Ueberschaar N, Ndejouong Ble S, Ding L, Maier A, Fiebig HH, Hertweck C.
Bioorg Med Chem Lett (2011) 21 : 5839 -5841
PubMed 21868221 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.37 6.98

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1834207 HYDRAZIDOMYCIN A 1 6.98
CHEMBL1834208 HYDRAZIDOMYCIN B 1 5.76

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1834207 HYDRAZIDOMYCIN A IC50 = 105.0 nM 6.98
CHEMBL1834208 HYDRAZIDOMYCIN B IC50 = 1730.0 nM 5.76