Assay Detail
ADMET
CHEMBL1924399
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Cytotoxicity against mouse NIH/3T3 cells
21
Total Activities
21
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Cell Type | NIH3T3 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Identification of small-molecule inhibitors of Trypansoma cruzi replication.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 4.27 | 4.71 |
| Activity | 5 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1794269 | — | — | 1 | 4.71 |
| CHEMBL1431319 | — | — | 1 | 4.38 |
| CHEMBL1705872 | — | — | 1 | 4.33 |
| CHEMBL1732272 | — | — | 1 | 4.29 |
| CHEMBL1703363 | — | — | 1 | 4.28 |
| CHEMBL1726621 | — | — | 1 | 4.21 |
| CHEMBL1708352 | — | — | 1 | 4.20 |
| CHEMBL1710224 | — | — | 1 | 4.19 |
| CHEMBL1433324 | — | — | 1 | 4.15 |
| CHEMBL1733202 | — | — | 1 | 4.13 |
| CHEMBL1619691 | — | — | 1 | 4.11 |
| CHEMBL1404654 | — | — | 1 | - |
| CHEMBL1415084 | — | — | 1 | - |
| CHEMBL1794268 | — | — | 1 | - |
| CHEMBL1794238 | — | — | 1 | - |
| CHEMBL1921857 | — | — | 1 | - |
| CHEMBL1328878 | — | — | 1 | - |
| CHEMBL1721356 | — | — | 1 | - |
| CHEMBL1193142 | — | — | 1 | - |
| CHEMBL1372575 | — | — | 1 | - |
| CHEMBL1459090 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1794269 | — | IC50 | = | 19500.0 | nM | 4.71 |
| CHEMBL1431319 | — | IC50 | = | 41700.0 | nM | 4.38 |
| CHEMBL1705872 | — | IC50 | = | 47000.0 | nM | 4.33 |
| CHEMBL1732272 | — | IC50 | = | 51000.0 | nM | 4.29 |
| CHEMBL1703363 | — | IC50 | = | 52700.0 | nM | 4.28 |
| CHEMBL1726621 | — | IC50 | = | 61600.0 | nM | 4.21 |
| CHEMBL1708352 | — | IC50 | = | 63300.0 | nM | 4.20 |
| CHEMBL1710224 | — | IC50 | = | 64700.0 | nM | 4.19 |
| CHEMBL1433324 | — | IC50 | = | 70300.0 | nM | 4.15 |
| CHEMBL1733202 | — | IC50 | = | 74300.0 | nM | 4.13 |
| CHEMBL1619691 | — | IC50 | = | 77300.0 | nM | 4.11 |
| CHEMBL1404654 | — | IC50 | - | — | - | |
| CHEMBL1415084 | — | Activity | - | — | - | |
| CHEMBL1794268 | — | IC50 | - | — | - | |
| CHEMBL1794238 | — | IC50 | - | — | - | |
| CHEMBL1921857 | — | IC50 | - | — | - | |
| CHEMBL1328878 | — | Activity | - | — | - | |
| CHEMBL1721356 | — | Activity | - | — | - | |
| CHEMBL1193142 | — | IC50 | = | 164000.0 | nM | - |
| CHEMBL1372575 | — | Activity | - | — | - | |
| CHEMBL1459090 | — | Activity | - | — | - |