Assay Detail
Binding
CHEMBL1937244
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Inhibition of FAAH
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Design, synthesis and evaluation of polar head group containing 2-keto-oxazole inhibitors of FAAH.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.39 | 6.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL90308 | — | — | 1 | 6.85 |
| CHEMBL93675 | — | — | 1 | 5.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL90308 | — | Ki | = | 140.0 | nM | 6.85 |
| CHEMBL93675 | — | Ki | = | 1200.0 | nM | 5.92 |