Assay Detail
Binding
CHEMBL1942537
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Inhibition of KDM4C
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Lysine demethylases inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 4.90 | 6.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1229308 | — | — | 1 | 6.00 |
| CHEMBL1938900 | — | — | 1 | 5.47 |
| CHEMBL1614745 | — | — | 1 | 4.10 |
| CHEMBL1615211 | — | — | 1 | 4.01 |
| CHEMBL90852 | N-OXALYLGLYCINE | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1229308 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL1938900 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL1614745 | — | IC50 | = | 79000.0 | nM | 4.10 |
| CHEMBL1615211 | — | IC50 | = | 97000.0 | nM | 4.01 |
| CHEMBL90852 | N-OXALYLGLYCINE | IC50 | = | 500000.0 | nM | - |