Assay Detail
Binding
CHEMBL1942540
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Inhibition of FIH
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Hypoxia-inducible factor 1-alpha inhibitor (CHEMBL5909) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Lysine demethylases inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.67 | 4.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1435274 | — | — | 1 | 4.68 |
| CHEMBL1938900 | — | — | 1 | 4.66 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1435274 | — | IC50 | = | 21000.0 | nM | 4.68 |
| CHEMBL1938900 | — | IC50 | = | 22000.0 | nM | 4.66 |